SCHEMBL17907932

SCHEMBL17907932

Cc1ccc2c(c1)cc1n2CC(=O)CC1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.41
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NOTUM Q6P988 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
F9 P00740 2/20 0.35
CYP2A6 P11509 2/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13279280 0.81 SIGMAR1 (0.42) SIGMAR1ALDH1A1KDM4EHSD17B10NOTUM
SCHEMBL17907930 0.81 HTR2A (0.48) ALDH1A1KDM4EHSD17B10NOTUMHTR2A
SCHEMBL17907920 0.80 HTR2A (0.51) ALDH1A1KDM4EHSD17B10SMN1; SMN2CYP2A6
SCHEMBL235219 0.78 NOTUM (0.59) SIGMAR1NOTUMHTR2AHTR2C
SCHEMBL9844702 0.77 NOTUM (0.62) SIGMAR1ALDH1A1KDM4ENPC1RAB9A
SCHEMBL17907965 0.71 HTR2A (0.48) NOTUMHTR2AHTR2CRXFP1
SCHEMBL9259274 0.69 KDM4E (0.39) SIGMAR1ALDH1A1KDM4ENPC1RAB9A
SCHEMBL17907947 0.68 ALDH1A1 (0.38) ALDH1A1NOTUML3MBTL1
SCHEMBL9259282 0.67 NOTUM (0.62) ALDH1A1KDM4EHSD17B10NOTUMSMN1; SMN2
SCHEMBL4705400 0.65 HTR2A (0.68) SIGMAR1KDM4EHSD17B10HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed