SCHEMBL180760

SCHEMBL180760

[C]1=CNc2ccccc2-c2ccccc21

nearest known ligand 0.30

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30
PDGFRA P16234 1/20 0.30
FER P16591 1/20 0.30
LTK P29376 1/20 0.30
CDK8 P49336 1/20 0.30
ACVR1 Q04771 1/20 0.30
LRRK2 Q5S007 1/20 0.30
DYRK1B Q9Y463 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4777381 0.64
SCHEMBL3942970 0.63 LRRK2 (0.45) MAOAMAOBPDGFRAFERLTK
SCHEMBL29353131 0.62 MAPT (0.41) MAOAMAOBPDGFRAFERLTK
SCHEMBL156862 0.62 MAPT (0.41) MAOAMAOBPDGFRAFERLTK
SCHEMBL1618358 0.61 MAOA (0.42) MAOAMAOBPDGFRAFERLTK
SCHEMBL102781 0.61 MEN1 (0.37) MAOAMAOBMAPT
SCHEMBL3021916 0.61
SCHEMBL181764 0.59 LRRK2 (0.59) MAOAMAOBPDGFRAFERLTK
SCHEMBL17816635 0.59 LRRK2 (0.59) MAOAMAOBPDGFRAFERLTK
SCHEMBL30462618 0.59 LRRK2 (0.59) MAOAMAOBPDGFRAFERLTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 718 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240199882-A1 THIENYL-DIBENZOAZEPINES AND THEIR DERIVATIVES AS DONORS FOR XANTHENE-BASED SHORT-WAVE INFRARED (SWIR) DYES MISSISSIPPI STATE UNIVERSITY (US) 2024-06-20 US claimed
WO-2024077223-A1 PROTEIN PHOSPHATASE 2A ACTIVATORS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2024-04-11 WO claimed
US-20220380357-A1 TETRAHYDROISOQUINOLINE COMPOUNDS ALLINKY BIOPHARMA (ES) 2022-12-01 US claimed
EP-3997086-A1 TETRAHYDROISOQUINOLINE COMPOUNDS Allinky Biopharma (ES) 2022-05-18 EP claimed
US-20210198235-A1 DERIVATIVES OF PIPERLONGUMINE AND USES THEREOF AURANSA INC. 2021-07-01 US claimed
WO-2021005165-A1 TETRAHYDROISOQUINOLINE COMPOUNDS ALLINKY BIOPHARMA (ES) 2021-01-14 WO claimed
WO-2019103897-A1 DERIVATIVES OF PIPERLONGUMINE AND USES THEREOF AURANSA INC. (US) 2019-05-31 WO claimed
US-8475686-B2 Bridged pyridoquinazoline or phenanthroline compounds and organic semiconducting material comprising that compound NOVALED AG (DE) 2013-07-02 US claimed
US-20120012794-A1 Bridged Pyridoquinazoline or Phenanthroline Compounds and Organic Semiconducting Material Comprising That Compound NOVALED AG (DE) 2012-01-19 US claimed
US-8084448-B2 Organic compounds NOVARTIS AG (CH) 2011-12-27 US claimed
US-5856331-A LYSOPHOSPHATIDIC ACYLTRANSFERASE INHIBITOR CELL THERAPEUTICS, INC. (US) 1999-01-05 US claimed
US-5576321-A ALKOXY-SUBSTITUTED INDOLES ELI LILLY AND COMPANY (US) 1996-11-19 US claimed
EP-0739203-A1 METHOD FOR TREATING DISEASES MEDIATED BY CELLULAR PROLIFERATION IN RESPONSE TO PDGF, EGF, FGF AND VEGF CELL THERAPEUTICS, INC. (US) 1996-10-30 EP claimed
EP-0728003-A1 METHOD FOR PREVENTING TISSUE INJURY FROM HYPOXIA CELL THERAPEUTICS, INC. (US) 1996-08-28 EP claimed
WO-1996022290-A1 COMPOUNDS HAVING EFFECTS ON SEROTONIN-RELATED SYSTEMS ELI LILLY AND COMPANY (US) 1996-07-25 WO claimed
EP-0722941-A2 Compounds having effects on serotonin-related systems ELI LILLY AND COMPANY (US) 1996-07-24 EP claimed
EP-0676958-A1 METHOD FOR INHIBITING INTRACELLULAR VIRAL REPLICATION CELL THERAPEUTICS, INC. (US) 1995-10-18 EP claimed
WO-1995019171-A1 METHOD FOR TREATING DISEASES MEDIATED BY CELLULAR PROLIFERATION IN RESPONSE TO PDGF, EGF, FGF AND VEGF CELL THERAPEUTICS, INC. (US) 1995-07-20 WO claimed
WO-1995013075-A1 METHOD FOR PREVENTING TISSUE INJURY FROM HYPOXIA CELL THERAPEUTICS, INC. (US) 1995-05-18 WO claimed
WO-1995012396-A1 METHOD FOR INHIBITING INTRACELLULAR VIRAL REPLICATION CELL THERAPEUTICS, INC. (US) 1995-05-11 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120012794-A1 Bridged Pyridoquinazoline or Phenanthroline Compounds and Organic Semiconducting Material Comprising That Compound PNPO, SDHB, PAH MAOA 218/4885MAOB 164/4885PDGFRA 3897/4885
US-20220380357-A1 TETRAHYDROISOQUINOLINE COMPOUNDS NDUFB5, GNAQ, SDHA MAOA 1131/4885MAOB 745/4885PDGFRA 3880/4885
US-20210198235-A1 DERIVATIVES OF PIPERLONGUMINE AND USES THEREOF THPO, PIR, PAK6 MAOA 3994/4885MAOB 3574/4885PDGFRA 37/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.