SCHEMBL18092205

SCHEMBL18092205

O=C(O)N1CCN(c2ccccc2C2CCCCCCC2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
PTGDR2 Q9Y5Y4 1/20 0.47
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
MAPT P10636 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
POLB P06746 1/20 0.44
TACR3 P29371 1/20 0.42
RAB9A P51151 2/20 0.42
NPY2R P49146 1/20 0.42
ALDH1A1 P00352 2/20 0.42
ALOX15 P16050 2/20 0.42
MAPK1 P28482 1/20 0.42
HTR1A P08908 1/20 0.42
ADRA1B P35368 1/20 0.42
NPC1 O15118 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18092179 0.83 RBP4 (0.46) TSHRNPY2RHTR1AADRA1BRBP4
SCHEMBL4851108 0.81 GPR119 (0.52) TSHRMEN1KMT2AMAPTALDH1A1
SCHEMBL23064544 0.81 PDCD1 (0.51) TSHRMEN1KMT2ANPSR1MAPK1
SCHEMBL27671027 0.80 HTR1A (0.42) TSHRMEN1KMT2AMAPTNPSR1
SCHEMBL23064565 0.79 PDCD1 (0.49) MAPTALDH1A1MAPK1HTR1AADRA1B
SCHEMBL8109274 0.78 ADRA2C (0.50) TSHRMEN1KMT2AMAPTPOLB
SCHEMBL2857040 0.76 AKR1C3 (0.64) MEN1KMT2AMAPTNPSR1SMN1; SMN2
SCHEMBL23064527 0.76 KEAP1 (0.47) MEN1KMT2AMAPTALDH1A1MAPK1
SCHEMBL23064465 0.76 KEAP1 (0.52) MAPTALDH1A1MAPK1HTR1AADRA1B
SCHEMBL4856101 0.75 ADRB1 (0.56) TSHRMAPTALDH1A1HTR1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1698620-B1 BENZENE COMPOUNDS DISUBSTITUTED WITH CYCLIC GROUPS AT THE 1- AND 2-POSITIONS EISAI R&D MAN CO LTD (JP) 2016-09-28 EP disclosed