SCHEMBL1811041

SCHEMBL1811041

O=C(O)c1cccc(NC(=O)c2ccccc2Cl)c1

nearest known ligand 0.81

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 2/20 0.81
KCNK9 Q9NPC2 2/20 0.81
SMO Q99835 2/20 0.68
MAPT P10636 2/20 0.67
PTGES O14684 1/20 0.64
NPC1 O15118 1/20 0.63
LMNA P02545 1/20 0.63
RAB9A P51151 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.63
KMT2A Q03164 4/20 0.63
MEN1 O00255 3/20 0.63
ALDH1A1 P00352 1/20 0.60
HPGD P15428 1/20 0.60
TP53 P04637 1/20 0.60
F2R P25116 1/20 0.59
POLB P06746 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2010680 0.98 KCNK3 (0.78) KCNK3KCNK9SMOMAPTPTGES
Ether SCHEMBL2011650 0.90 KCNK3 (0.66) KCNK3KCNK9SMOMAPTPTGES
SCHEMBL2005896 0.88 KCNK3 (0.76) KCNK3KCNK9SMOMAPTPTGES
SCHEMBL2058337 0.86 ALDH1A1 (0.71) KCNK3KCNK9NPC1LMNARAB9A
Hydrochloric Acid SCHEMBL2105080 0.84 MEN1 (0.64) KCNK3KCNK9MAPTNPC1LMNA
SCHEMBL1813249 0.84 RAB9A (0.81) KCNK3KCNK9MAPTPTGESNPC1
SCHEMBL1203522 0.84 SMO (0.80) KCNK3KCNK9SMOMAPTNPC1
SCHEMBL19491387 0.83 KCNK3 (0.78) KCNK3KCNK9SMOMAPTNPC1
Hydrochloric Acid SCHEMBL2103616 0.83 NPC1 (0.61) KCNK3KCNK9NPC1LMNARAB9A
SCHEMBL15778718 0.83 FADS1 (0.74) KCNK3KCNK9SMOMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12310944-B2 Selective butyrylcholinesterase inhibitor or pharmaceutically acceptable salt thereof, preparation method and use thereof CHINA PHARMACEUTICAL UNIVERSITY (CN) 2025-05-27 US disclosed
US-20230165833-A1 Selective Butyrylcholinesterase Inhibitor or Pharmaceutically Acceptable Salt Thereof, Preparation Method and Use Thereof CHINA PHARMACEUTICAL UNIVERSITY (CN) 2023-06-01 US disclosed
WO-2021042410-A1 SELECTIVE BUTYRYLCHOLINESTERASE INHIBITOR OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 中国药科大学 2021-03-11 WO disclosed
CN-110627767-B Selective butyrylcholinesterase inhibitor or pharmaceutically acceptable salt thereof, preparation method and application thereof 中国药科大学 2020-08-25 CN disclosed
EP-2535327-A1 Insecticidal 3-acylaminobenzanilides Bayer CropScience AG (DE) 2012-12-19 EP disclosed
EP-2535327-A1 Insecticidal 3-acylaminobenzanilides Bayer CropScience AG (DE) 2012-12-19 EP disclosed
US-8207219-B2 Ion channel modulating activity I CARDIOME PHARMA CORP. (CA) 2012-06-26 US disclosed
US-20120095073-A1 ION CHANNEL MODULATING ACTIVITY II CARDIOME PHARMA CORP. (CA) 2012-04-19 US disclosed
CN-102177135-A Acylaminobenzamide derivatives BAYER CROPSCIENCE AG 2011-09-07 CN disclosed
US-20110201603-A1 Novel Acylaminobenzamide Derivatives BAYER CROPSCIENCE AG (DE) 2011-08-18 US disclosed
WO-2005018635-A2 ION CHANNEL MODULATING ACTIVITY I CARDIOME PHARMA CORP. (CA) 2005-03-03 WO disclosed
US-20030186998-A1 Methods for treatment of disorders of cardiac contractility JOHN HOPKINS UNIVERSITY 2003-10-02 US disclosed
US-6569862-B1 Adminstering xanthine oxidase inhibitor such as allopurinol JOHNS HOPKINS UNIVERSITY 2003-05-27 US disclosed
EP-1044002-A4 METHODS FOR TREATMENT OF DISORDERS OF CARDIAC CONTRACTILITY UNIV JOHNS HOPKINS (US) 2003-05-02 EP disclosed
US-6191136-B1 ADMINISTERING XANTHINE OXIDASE INHIBITOR JOHNS HOPKINS UNIVERSITY 2001-02-20 US disclosed
EP-1044002-A1 METHODS FOR TREATMENT OF DISORDERS OF CARDIAC CONTRACTILITY JOHNS HOPKINS UNIVERSITY (US) 2000-10-18 EP disclosed
WO-1999024038-A1 METHODS FOR TREATMENT OF DISORDERS OF CARDIAC CONTRACTILITY JOHNS HOPKINS UNIVERSITY (US) 1999-05-20 WO disclosed
US-5674887-A Prevention of bone resorption ELI LILLY AND COMPANY (US) 1997-10-07 US disclosed
US-5436258-A Prevention of bone resorption ELI LILLY AND COMPANY (US) 1995-07-25 US disclosed
EP-0587378-A1 Prevention of bone resorption ELI LILLY AND COMPANY (US) 1994-03-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030186998-A1 Methods for treatment of disorders of cardiac contractility TNNI3, TNNT2, RYR2 KCNK3 745/4885KCNK9 1465/4885SMO 3822/4885
US-20110201603-A1 Novel Acylaminobenzamide Derivatives KCNB1, KCNA5, KCNA7 KCNK3 174/4885KCNK9 461/4885SMO 4590/4885
US-20230165833-A1 Selective Butyrylcholinesterase Inhibitor or Pharmaceutically Acceptable Salt Thereof, Preparation Method and Use Thereof BCHE, ACHE, BACE1 KCNK3 1980/4885KCNK9 545/4885SMO 2084/4885
US-12310944-B2 Selective butyrylcholinesterase inhibitor or pharmaceutically acceptable salt thereof, preparation method and use thereof BCHE, ACHE, BACE1 KCNK3 2135/4885KCNK9 679/4885SMO 2236/4885
US-20120095073-A1 ION CHANNEL MODULATING ACTIVITY II KCNH1, KCNN3, KCNJ2 KCNK3 77/4885KCNK9 83/4885SMO 4600/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.