SCHEMBL18315551

SCHEMBL18315551

O=C(O)NC1CC2(C1)CC(C(=O)Nc1ccc3[nH]nnc3c1)C2

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.48
ATXN2 Q99700 1/20 0.48
POLB P06746 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
ULK1 O75385 6/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PDPK1 O15530 3/20 0.36
ITK Q08881 3/20 0.34
BRD4 O60885 1/20 0.34
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL16616663 0.81 ULK1 (0.41) ENPP2ATXN2POLBMAOAMAOB
SCHEMBL15553437 0.81 ENPP2 (0.77) ENPP2ATXN2
SCHEMBL18315523 0.76 ENPP2 (0.49) ENPP2ATXN2POLBULK1L3MBTL1
SCHEMBL142543 0.75 ULK1 (0.56) POLBULK1L3MBTL1PDPK1
SCHEMBL16070870 0.71 SMN1; SMN2 (0.46) POLB
SCHEMBL16069965 0.69 TERT (0.48)
SCHEMBL1247686 0.69 ROCK2 (0.55) POLBMAOAMAOBKDM4ETP53
SCHEMBL1156215 0.69 PEPD (0.42) PDPK1ROCK2ROCK1MAPT
SCHEMBL9172845 0.68 ROCK2 (0.54) POLBMAOAMAOBKDM4ETP53
SCHEMBL14360693 0.68 CA2 (0.46) POLBKDM4ETP53ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2861566-B1 NEW DIAZASPIROCYCLOALKANE AND AZASPIROCYCLOALKANE HOFFMANN LA ROCHE (CH) 2016-12-21 EP claimed