SCHEMBL1831667

SCHEMBL1831667

CNC(=O)OC(c1cn(S(=O)(=O)c2ccc(OC)cn2)c(-c2cccnc2F)c1F)C(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 2/20 0.33
GSK3B P49841 1/20 0.33
GRM4 Q14833 1/20 0.32
MMP2 P08253 2/20 0.32
MMP9 P14780 2/20 0.32
MMP8 P22894 2/20 0.32
MMP13 P45452 2/20 0.32
KAT8 Q9H7Z6 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1835872 0.91 GRM4 (0.31) GRM4
SCHEMBL1834071 0.89 NFE2L2 (0.33) NFE2L2GSK3BMMP2MMP9MMP8
SCHEMBL4415071 0.85 ALDH1A1 (0.30) ALDH1A1
SCHEMBL4424412 0.84 SLC40A1 (0.31)
SCHEMBL1837632 0.83 PTGS2 (0.30)
SCHEMBL1831693 0.83
SCHEMBL4425554 0.83 RORC (0.33)
SCHEMBL2412509 0.83
SCHEMBL1832698 0.82 RORC (0.32)
SCHEMBL2408490 0.82 HTR6 (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318390-A1 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2011-05-11 EP disclosed
WO-2010024451-A1 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-03-04 WO disclosed