SCHEMBL19009080

SCHEMBL19009080

COc1cccc(N(C)C(C)C)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.49
SLC6A4 P31645 1/20 0.49
MTNR1A P48039 6/20 0.48
MTNR1B P49286 6/20 0.48
TAAR1 Q96RJ0 3/20 0.47
HSD17B2 P37059 2/20 0.45
ALOX15 P16050 1/20 0.45
HSD17B1 P14061 1/20 0.45
ACHE P22303 1/20 0.45
AOC3 Q16853 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12369341 0.83 RXRA (0.41) MTNR1AMTNR1BACHECA2ALDH1A1
SCHEMBL26042904 0.82 TAAR1 (0.51) SLC6A2SLC6A4MTNR1AMTNR1BTAAR1
SCHEMBL14940633 0.82 TAAR1 (0.48) MTNR1AMTNR1BTAAR1HSD17B2ALOX15
SCHEMBL24300289 0.80 TP53 (0.49) MTNR1AMTNR1BALOX15ALDH1A1CYP3A4
SCHEMBL1134082 0.79 MTNR1A (0.61) MTNR1AMTNR1BHSD17B2ALOX15HSD17B1
SCHEMBL29636366 0.79 ACHE (0.52) MTNR1AMTNR1BHSD17B2ALOX15HSD17B1
SCHEMBL30054343 0.79 MTNR1A (0.61) MTNR1AMTNR1BHSD17B2ALOX15HSD17B1
SCHEMBL820669 0.79 ACHE (0.52) MTNR1AMTNR1BHSD17B2ALOX15HSD17B1
SCHEMBL19009081 0.79 ALDH1A1 (0.50) ALDH1A1CYP3A4
SCHEMBL24300188 0.79 GRM2 (0.45) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102285904-B Method for preparing rivastigmine CHENGDU INST BIOLOGY CAS 2013-06-05 CN claimed
CN-102285904-A Method for preparing rivastigmine 2011-12-21 CN claimed
US-20240018118-A1 TRICYCLIC COMPOUNDS TO DEGRADE NEOSUBSTRATES FOR MEDICAL THERAPY C 4 Therapeutics, Inc. (US) 2024-01-18 US disclosed
US-10889556-B2 Compositions and methods for inhibiting influenza RNA polymerase PA endonuclease THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-01-12 US disclosed
US-20190106398-A1 COMPOSITIONS AND METHODS FOR INHIBITING INFLUENZA RNA POLYMERASE PA ENDONUCLEASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2019-04-11 US disclosed
CN-108822000-A A kind of method of reduction amination synthesis (S)-Rivastigmine 山东师范大学 2018-11-16 CN disclosed
US-20170174639-A1 EIS INHIBITORS UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION 2017-06-22 US disclosed
CN-102285904-B Method for preparing rivastigmine CHENGDU INST BIOLOGY CAS 2013-06-05 CN disclosed
CN-102285904-A Method for preparing rivastigmine 2011-12-21 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190106398-A1 COMPOSITIONS AND METHODS FOR INHIBITING INFLUENZA RNA POLYMERASE PA ENDONUCLEASE POLRMT, RNASE1, POLM SLC6A2 4258/4885SLC6A4 4358/4885MTNR1A 2103/4885
US-20170174639-A1 EIS INHIBITORS ABCC1, ATP5ME, ABCG2 SLC6A2 1634/4885SLC6A4 3058/4885MTNR1A 4222/4885
US-20240018118-A1 TRICYCLIC COMPOUNDS TO DEGRADE NEOSUBSTRATES FOR MEDICAL THERAPY NFATC1, CTSS, MMP12 SLC6A2 2569/4885SLC6A4 2521/4885MTNR1A 2382/4885
US-10889556-B2 Compositions and methods for inhibiting influenza RNA polymerase PA endonuclease POLRMT, RNASE1, POLM SLC6A2 4258/4885SLC6A4 4358/4885MTNR1A 2103/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.