SCHEMBL19085975

SCHEMBL19085975

CC[C@@H](NC(=O)c1cc2cn[nH]c2cc1OC)C(=O)N1CCc2sc(C(=O)NCc3cc(F)ccc3C)cc2C1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 9/20 0.37
WDR77 Q9BQA1 9/20 0.37
USP2 O75604 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HCRTR2 O43614 3/20 0.33
GRK2 P25098 1/20 0.33
GRK5 P34947 1/20 0.33
ROCK1 Q13464 1/20 0.33
GRK1 Q15835 1/20 0.33
KDM1A O60341 3/20 0.33
HDAC6 Q9UBN7 3/20 0.33
MAP3K5 Q99683 1/20 0.33
HCRTR1 O43613 1/20 0.33
ROCK2 O75116 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19085997 0.89 PRMT5 (0.40) PRMT5WDR77ROCK1ROCK2
SCHEMBL19085992 0.89 PRMT5 (0.40) PRMT5WDR77ROCK1ROCK2
SCHEMBL19085986 0.85 PRMT5 (0.39) PRMT5WDR77HCRTR2ROCK1HCRTR1
SCHEMBL19085988 0.84 HCRTR2 (0.40) PRMT5WDR77HCRTR2HCRTR1
SCHEMBL19086010 0.84 PRMT5 (0.36) PRMT5WDR77USP2HCRTR2KDM1A
SCHEMBL19085979 0.82 MAOB (0.41) PRMT5WDR77ROCK1KDM1AHDAC6
SCHEMBL19086041 0.81 ROCK2 (0.40) PRMT5WDR77USP2HCRTR2ROCK1
SCHEMBL19085982 0.80 KDM4E (0.39) PRMT5WDR77HCRTR2ROCK1KDM1A
SCHEMBL19085980 0.80 PRMT5 (0.40) PRMT5WDR77ROCK1HDAC6ROCK2
SCHEMBL19086260 0.80 METTL3 (0.38) PRMT5WDR77ROCK1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed