SCHEMBL191625

SCHEMBL191625

CC1CN(C(c2ccccc2)(c2ccccc2)c2ccccc2)CCN1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.39
CYP2B6 P20813 1/20 0.37
KDM4E B2RXH2 1/20 0.36
KHK P50053 2/20 0.36
SIGMAR1 Q99720 2/20 0.34
BIRC2 Q13490 2/20 0.34
XIAP P98170 1/20 0.34
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
ATM Q13315 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
NFKB1 P19838 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL236732 1.00 HRH4 (0.39) HRH4CYP2B6KDM4EKHKSIGMAR1
SCHEMBL191624 1.00 HRH4 (0.39) HRH4CYP2B6KDM4EKHKSIGMAR1
SCHEMBL27927305 0.78 LTA4H (0.30) CYP2B6
SCHEMBL334587 0.78 MAPT (0.40) HTR2AHTR2CHTR2BLMNA
SCHEMBL30067321 0.77 LTA4H (0.41)
SCHEMBL30067331 0.77 LTA4H (0.41)
SCHEMBL1206174 0.77 LTA4H (0.41)
SCHEMBL10362321 0.75 EIF2AK4 (0.35) HRH4LMNA
SCHEMBL5732869 0.75 LTA4H (0.34) SIGMAR1HTR2AHTR2CHTR2BHRH3
SCHEMBL18803696 0.75 CHRM3 (0.43) CYP2B6SIGMAR1LMNAATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104046246-B The chemical-mechanical planarization of tungsten-containing substrate 气体产品与化学公司 2016-06-15 CN claimed
US-20140273458-A1 Chemical Mechanical Planarization for Tungsten-Containing Substrates AIR PRODUCTS AND CHEMICALS, INC. (US) 2014-09-18 US claimed
EP-2779217-A2 Chemical mechanical planarization for tungsten-containing substrates AIR PRODUCTS AND CHEMICALS, INC. (US) 2014-09-17 EP claimed
US-7129354-B2 Process for the preparation of stable acid addition salt of 2,3-disubstituted pyrazine compounds BIOVITRUM AB (SE) 2006-10-31 US claimed
EP-1529043-B1 Process for the preparation of 2-methyl piperazine derivatives. BIOVITRUM AB (SE) 2006-08-02 EP claimed
US-20060142578-A1 Novel process BIOVITRUM AB, A SWEDEN CORPORATION 2006-06-29 US claimed
EP-1529043-A1 NOVEL PROCESS Biovitrum AB (SE) 2005-05-11 EP claimed
US-20040038981-A1 Novel Process PROXIMAGEN NEUROSCIENCE PLC (GB) 2004-02-26 US claimed
WO-2004000829-A1 NOVEL PROCESS BIOVITRUM AB (SE) 2003-12-31 WO claimed
EP-3728267-B1 TRICYCLIC INHIBITORS OF THE BCL6 BTB DOMAIN PROTEIN-PROTEIN INTERACTION AND USES THEREOF ONTARIO INSTITUTE FOR CANCER RES OICR (CA) 2023-09-13 EP disclosed
US-11242351-B2 Tricyclic inhibitors of the BCL6 BTB domain protein-protein interaction and uses thereof ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR) (CA) 2022-02-08 US disclosed
US-20210053978-A1 TRICYCLIC INHIBITORS OF THE BCL6 BTB DOMAIN PROTEIN-PROTEIN INTERACTION AND USES THEREOF ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR) (CA) 2021-02-25 US disclosed
EP-3728267-A1 TRICYCLIC INHIBITORS OF THE BCL6 BTB DOMAIN PROTEIN-PROTEIN INTERACTION AND USES THEREOF Ontario Institute for Cancer Research (OICR) (CA) 2020-10-28 EP disclosed
US-9943519-B2 Pharmaceutical compounds GENENTECH, INC. (US) 2018-04-17 US disclosed
US-20040242554-A1 CERTAIN ARYLALIPHATIC AND HETEROARYL-ALIPHATIC PIPERAZINYL PYRAZINES AND THEIR USE IN THE TREATMENT OF SEROTONIN-RELATED DISEASES BIOVITRUM, AB, A STOCKHOLM, SWEDEN CORPORATION 2004-12-02 US disclosed
US-20040038981-A1 Novel Process PROXIMAGEN NEUROSCIENCE PLC (GB) 2004-02-26 US disclosed
WO-2004000829-A1 NOVEL PROCESS BIOVITRUM AB (SE) 2003-12-31 WO disclosed
US-20030232814-A1 Novel compounds and their use BIOVITRUM AB (PUBL) (SE) 2003-12-18 US disclosed
US-20030092694-A1 Certain arylaliphatic and heteroaryl-aliphatic piperazinyl pyrazines and their use in the treatment of serotonin-related diseases BIOVITRUM, AB, A STOCKHOLM, SWEDEN CORPORATION 2003-05-15 US disclosed
US-6465467-B1 DISEASES RELATED TO THE 5-HT2C RECEPTOR, ESPECIALLY EATING, MEMORY, MOOD, URINARY AND ANXIETY DISORDERS, SCHIZOPHRENIA, PAIN, SEXUAL DYSFUNCTIONS BIOVITRUM AB (SE) 2002-10-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030092694-A1 Certain arylaliphatic and heteroaryl-aliphatic piperazinyl pyrazines and their use in the treatment of serotonin-related diseases HTR2C, HTR3C, HTR2A HRH4 219/4885CYP2B6 128/4885KDM4E 2431/4885
US-20040242554-A1 CERTAIN ARYLALIPHATIC AND HETEROARYL-ALIPHATIC PIPERAZINYL PYRAZINES AND THEIR USE IN THE TREATMENT OF SEROTONIN-RELATED DISEASES HTR2C, HTR3C, HTR2A HRH4 213/4885CYP2B6 122/4885KDM4E 2230/4885
US-20210053978-A1 TRICYCLIC INHIBITORS OF THE BCL6 BTB DOMAIN PROTEIN-PROTEIN INTERACTION AND USES THEREOF BCL6, BCL6B, BCL3 HRH4 4545/4885CYP2B6 3153/4885KDM4E 434/4885
US-20030232814-A1 Novel compounds and their use GPR119, FABP4, MC4R HRH4 553/4885CYP2B6 169/4885KDM4E 1929/4885
US-11242351-B2 Tricyclic inhibitors of the BCL6 BTB domain protein-protein interaction and uses thereof BCL6, BCL6B, BCL3 HRH4 4545/4885CYP2B6 3153/4885KDM4E 434/4885
US-20040038981-A1 Novel Process HTR1A, TPH1, HTR1B HRH4 28/4885CYP2B6 54/4885KDM4E 3310/4885
US-20060142578-A1 Novel process HTR1A, TPH1, HTR5A HRH4 17/4885CYP2B6 87/4885KDM4E 4340/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.