SCHEMBL19557296

SCHEMBL19557296

C[Si](C)(c1ccccc1)c1cc2ccccc2s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.43
ADRB2 P07550 1/20 0.43
ASIC3 Q9UHC3 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
BCL2L1 Q07817 1/20 0.42
AGXT P21549 1/20 0.40
MGLL Q99685 1/20 0.39
CA12 O43570 2/20 0.39
CA9 Q16790 2/20 0.39
CA2 P00918 2/20 0.39
CA1 P00915 1/20 0.39
CA4 P22748 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
ADRA1D P25100 2/20 0.36
GRM5 P41594 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30444190 1.00 CYP2A6 (0.43) CYP2A6ADRB2ASIC3LOXL2BCL2L1
SCHEMBL17010954 0.84 ESR1 (0.43) ESR1ESR2LMNA
SCHEMBL28514083 0.81 BCL2L1 (0.44) CYP2A6ADRB2ASIC3LOXL2BCL2L1
SCHEMBL31141892 0.81 BCL2L1 (0.44) CYP2A6ADRB2ASIC3LOXL2BCL2L1
SCHEMBL6596113 0.80 CYP2A6 (0.48) CYP2A6ADRB2ASIC3LOXL2BCL2L1
SCHEMBL17856939 0.72 CYP2A6 (0.44) CYP2A6ADRB2ASIC3LOXL2BCL2L1
SCHEMBL30444116 0.72 CYP2A6 (0.44) CYP2A6ADRB2ASIC3LOXL2BCL2L1
SCHEMBL18271669 0.69 MGLL (0.42) CYP2A6ADRB2ASIC3LOXL2BCL2L1
SCHEMBL63526 0.67 ESR1 (0.70) CA4ESR1ESR2LMNAALOX12
SCHEMBL12921500 0.67 L3MBTL1 (0.44) ASIC3GAAALOX15CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11753421-B2 Silylated derivatives of aromatic heterocycles CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2023-09-12 US disclosed
US-11753421-B2 Silylated derivatives of aromatic heterocycles CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2023-09-12 US disclosed
EP-3705482-B1 SILYLATION OF AROMATIC HETEROCYCLES BY EARTH ABUNDANT TRANSITION-METAL-FREE CATALYSTS CALIFORNIA INST OF TECHN (US) 2023-02-22 EP disclosed
US-20220185828-A1 Silylated Derivatives Of Aromatic Heterocycles CALIFORNIA INSTITUTE OF TECHNOLOGY 2022-06-16 US disclosed
US-20220162236-A1 SILYLATIONS OF AROMATIC SUBSTRATES WITH BASE-ACTIVATED ORGANOSILANES CALIFORNIA INSTITUTE OF TECHNOLOGY 2022-05-26 US disclosed
US-11312733-B2 Silylated derivatives of aromatic heterocycles CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-04-26 US disclosed
US-11230520-B2 Silylations of aromatic substrates with base-activated organosilanes CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-01-25 US disclosed
US-20210122701-A1 SILYLATIONS OF AROMATIC SUBSTRATES WITH BASE-ACTIVATED ORGANOSILANES CALIFORNIA INSTITUTE OF TECHNOLOGY 2021-04-29 US disclosed
US-10927065-B2 Silylations of aromatic substrates with base-activated organosilanes CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2021-02-23 US disclosed
US-20180155271-A1 SILYLATIONS OF AROMATIC SUBSTRATES WITH BASE-ACTIVATED ORGANOSILANES CALIFORNIA INSTITUTE OF TECHNOLOGY 2018-06-07 US disclosed
US-20180155271-A1 SILYLATIONS OF AROMATIC SUBSTRATES WITH BASE-ACTIVATED ORGANOSILANES CALIFORNIA INSTITUTE OF TECHNOLOGY 2018-06-07 US disclosed
US-9908840-B2 Reactions of aromatic substrates with base-activated hydrosilanes-silylations and reductive cleavage CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-03-06 US disclosed
US-9908840-B2 Reactions of aromatic substrates with base-activated hydrosilanes-silylations and reductive cleavage CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-03-06 US disclosed
US-20180057514-A1 SILYLATION OF AROMATIC HETEROCYCLES BY EARTH ABUNDANT TRANSITION-METAL-FREE CATALYSTS CALIFORNIA INSTITUTE OF TECHNOLOGY 2018-03-01 US disclosed
US-9809607-B2 Silylation of aromatic heterocycles by earth abundant transition-metal-free catalysts CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2017-11-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10927065-B2 Silylations of aromatic substrates with base-activated organosilanes TYR, DDC, TPST2 CYP2A6 684/4885ADRB2 3192/4885ASIC3 2608/4885
US-20180155271-A1 SILYLATIONS OF AROMATIC SUBSTRATES WITH BASE-ACTIVATED ORGANOSILANES TYR, DDC, TPST2 CYP2A6 684/4885ADRB2 3192/4885ASIC3 2608/4885
US-11230520-B2 Silylations of aromatic substrates with base-activated organosilanes TYR, DDC, TPST2 CYP2A6 684/4885ADRB2 3192/4885ASIC3 2608/4885
US-11312733-B2 Silylated derivatives of aromatic heterocycles KCNH1, KCNH3, HNRNPH3 CYP2A6 2952/4885ADRB2 1447/4885ASIC3 895/4885
US-20220162236-A1 SILYLATIONS OF AROMATIC SUBSTRATES WITH BASE-ACTIVATED ORGANOSILANES TYR, DDC, TPST2 CYP2A6 684/4885ADRB2 3192/4885ASIC3 2608/4885
US-20180057514-A1 SILYLATION OF AROMATIC HETEROCYCLES BY EARTH ABUNDANT TRANSITION-METAL-FREE CATALYSTS TEC, AURKA, TYR CYP2A6 1097/4885ADRB2 2998/4885ASIC3 1561/4885
US-11753421-B2 Silylated derivatives of aromatic heterocycles KCNH1, KCNH3, HNRNPH3 CYP2A6 2952/4885ADRB2 1447/4885ASIC3 895/4885
US-20220185828-A1 Silylated Derivatives Of Aromatic Heterocycles KCNH1, KCNH3, HNRNPH3 CYP2A6 2952/4885ADRB2 1447/4885ASIC3 895/4885
US-20210122701-A1 SILYLATIONS OF AROMATIC SUBSTRATES WITH BASE-ACTIVATED ORGANOSILANES TYR, DDC, TPST2 CYP2A6 684/4885ADRB2 3192/4885ASIC3 2608/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.