SCHEMBL19682469

SCHEMBL19682469

O=C1NC(=O)c2cc(S(=O)(=O)Cl)ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPOX P50336 1/20 0.53
ATIC P31939 1/20 0.51
TDP1 Q9NUW8 2/20 0.47
CYP3A4 P08684 1/20 0.47
MAOA P21397 7/20 0.43
MAOB P27338 7/20 0.43
GSK3B P49841 1/20 0.43
CASP3 P42574 2/20 0.42
CASP2 P42575 1/20 0.42
CASP7 P55210 1/20 0.42
CASP6 P55212 1/20 0.42
CASP8 Q14790 1/20 0.42
GRM5 P41594 3/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
KLK7 P49862 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15698878 0.83 PPOX (0.52) PPOXATICTDP1CYP3A4MAOA
SCHEMBL11127435 0.80 CA1 (0.62) PPOXATICTDP1CYP3A4GSK3B
SCHEMBL2896434 0.80 PPOX (0.48) PPOXATICTDP1CYP3A4MAOA
SCHEMBL2265043 0.79 PKM (0.47) TDP1CYP3A4MAOAMAOBALDH1A1
SCHEMBL55616 0.79 PKM (0.47) TDP1CYP3A4MAOAMAOBALDH1A1
SCHEMBL2264974 0.79 PKM (0.48) TDP1MAOAMAOBALDH1A1HSD17B10
SCHEMBL31121547 0.79 PKM (0.47) TDP1CYP3A4MAOAMAOBALDH1A1
SCHEMBL30555218 0.77 CA12 (0.69) MAOAMAOBCASP3CASP7CA12
SCHEMBL565240 0.77 CA12 (0.69) MAOAMAOBCASP3CASP7CA12
SCHEMBL3291294 0.76 ALDH1A1 (0.47) TDP1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10889555-B2 Sulfonamide compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2021-01-12 US disclosed
US-20200405697-A1 Antitumor Agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-31 US disclosed
US-20200399235-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-24 US disclosed
EP-3718545-A1 ANTITUMOR AGENT Taiho Pharmaceutical Co., Ltd. (JP) 2020-10-07 EP disclosed
US-20200157066-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-05-21 US disclosed
EP-3466934-A1 SULFONAMIDE COMPOUND OR SALT THEREOF Taiho Pharmaceutical Co., Ltd. (JP) 2019-04-10 EP disclosed
WO-2017209155-A1 SULFONAMIDE COMPOUND OR SALT THEREOF 大鵬薬品工業株式会社 2017-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200399235-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 PPOX 3717/4885ATIC 1651/4885TDP1 2190/4885
US-20200157066-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 PPOX 3717/4885ATIC 1651/4885TDP1 2190/4885
US-10889555-B2 Sulfonamide compound or salt thereof RNASEH1, SNRPA1, RRM2 PPOX 3717/4885ATIC 1651/4885TDP1 2190/4885
US-20200405697-A1 Antitumor Agent HNRNPR, RRM2, RRM2B PPOX 3566/4885ATIC 2632/4885TDP1 2642/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.