SCHEMBL198507

SCHEMBL198507

C[C@H](C#N)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
TRPA1 O75762 1/20 0.52
MIF P14174 2/20 0.41
TAAR1 Q96RJ0 3/20 0.41
KDM4E B2RXH2 2/20 0.39
ADRA2A P08913 1/20 0.39
ADRA2C P18825 1/20 0.39
CYP2D6 P10635 1/20 0.39
LMNA P02545 1/20 0.39
HIF1A Q16665 1/20 0.39
ALDH1A1 P00352 4/20 0.39
MAPT P10636 1/20 0.39
HSD17B10 Q99714 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C1 Q04828 1/20 0.39
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
RAB9A P51151 1/20 0.38
ALOX5 P09917 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28208618 1.00 TSHR (0.52) TSHRTRPA1MIFTAAR1KDM4E
SCHEMBL7039581 1.00 TSHR (0.52) TSHRTRPA1MIFTAAR1KDM4E
SCHEMBL156029 1.00 TSHR (0.52) TSHRTRPA1MIFTAAR1KDM4E
SCHEMBL909548 0.97 TRPA1 (0.50) TSHRTRPA1MIFTAAR1KDM4E
SCHEMBL954845 0.86 PTGS2 (0.48) TSHRTRPA1ALDH1A1
SCHEMBL6565095 0.86 ESR1 (0.43) TSHRTRPA1ALDH1A1AKR1C3AKR1C1
SCHEMBL11144946 0.84 PBRM1 (0.45) TSHRTRPA1TAAR1KDM4EADRA2A
SCHEMBL5324135 0.84 PTGS2 (0.56) TSHRKDM4ECYP2D6LMNAHIF1A
SCHEMBL28153074 0.84 TRPA1 (0.39) TSHRTRPA1TAAR1KDM4ELMNA
SCHEMBL9079901 0.81 CTSK (0.48) TSHRTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2327766-B1 Nitrilases BASF ENZYMES LLC (US) 2015-12-02 EP claimed
EP-2319919-B1 Nitrilases BASF ENZYMES LLC (US) 2015-08-12 EP claimed
EP-2327767-B1 Nitrilases BASF ENZYMES LLC (US) 2015-04-29 EP claimed
EP-2327765-B1 Nitrilases BASF ENZYMES LLC (US) 2015-04-01 EP claimed
US-20130177949-A1 NITRILASES VERENIUM CORPORATION (US) 2013-07-11 US claimed
EP-2327767-A1 Nitrilases Verenium Corporation (US) 2011-06-01 EP claimed
EP-2327766-A1 Nitrilases Verenium Corporation (US) 2011-06-01 EP claimed
EP-2327765-A1 Nitrilases Verenium Corporation (US) 2011-06-01 EP claimed
EP-2319919-A1 Nitrilases Verenium Corporation (US) 2011-05-11 EP claimed
EP-2039762-A2 Nitralases Verenium Corporation (US) 2009-03-25 EP claimed
US-20030124698-A1 Which stereoselectively hydrolyze nitrites or cyanohydrins into acids and ammonia DIVERSA CORPORATION 2003-07-03 US claimed
WO-2023150374-A1 INDUCERS OF KLF2 AND METHODS OF USE THEREOF RIPARIAN PHARMACEUTICALS, INC. (US) 2023-08-10 WO disclosed
WO-2021212039-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. (US) 2021-10-21 WO disclosed
CN-109486897-A A kind of method that stereoselectivity enzymatic hydrolysis splits 2- phenylpropionic acid enantiomer 湖南理工学院 2019-03-19 CN disclosed
US-20180194747-A1 Heterocyclic compounds, medicaments containing said compounds, use thereof and processes for the preparation thereof BOEHRINGER INGELHEIM INT (DE) 2018-07-12 US disclosed
US-20040002147-A1 Nitrilases DIVERSA CORPORATION 2004-01-01 US disclosed
WO-2003097810-A2 NITRILASES, NUCLEIC ACIDS ENCODING THEM AND METHODS FOR MAKING AND USING THEM DIVERSA CORPORATION (US) 2003-11-27 WO disclosed
US-20030124698-A1 Which stereoselectively hydrolyze nitrites or cyanohydrins into acids and ammonia DIVERSA CORPORATION 2003-07-03 US disclosed
US-5258305-A Manufacture of optically active 2-phenylpropionic acid and 2-phenylpropionamide from the nitrile using Rhodococcus equi NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1993-11-02 US disclosed
US-5258305-A Manufacture of optically active 2-phenylpropionic acid and 2-phenylpropionamide from the nitrile using Rhodococcus equi NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1993-11-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180194747-A1 Heterocyclic compounds, medicaments containing said compounds, use thereof and processes for the preparation thereof SCNN1B, SCNN1A, TRPM5 TSHR 4441/4885TRPA1 9/4885MIF 2672/4885
US-20040002147-A1 Nitrilases RNGTT, DNTT, NOP2 TSHR 4001/4885TRPA1 2778/4885MIF 3707/4885
US-20030124698-A1 Which stereoselectively hydrolyze nitrites or cyanohydrins into acids and ammonia NIT2, DNPH1, ASNS TSHR 4562/4885TRPA1 2608/4885MIF 3211/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.