SCHEMBL19860111

SCHEMBL19860111

O=C(CNCc1ccccn1)Nc1ccc2cnccc2c1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.55
KDM4E B2RXH2 1/20 0.55
IMPDH2 P12268 3/20 0.54
ALDH1A1 P00352 1/20 0.52
GAA P10253 1/20 0.52
PRMT3 O60678 4/20 0.51
NTRK1 P04629 2/20 0.48
NTRK3 Q16288 1/20 0.48
ROCK2 O75116 4/20 0.48
ROCK1 Q13464 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2162616 0.85 IMPDH2 (0.70) NOTUMKDM4EIMPDH2ALDH1A1GAA
SCHEMBL19860124 0.82 IMPDH2 (0.59) NOTUMKDM4EIMPDH2ALDH1A1PRMT3
SCHEMBL19860110 0.81 IMPDH2 (0.59) NOTUMIMPDH2PRMT3ROCK2ROCK1
SCHEMBL19860043 0.81 NOTUM (0.63) NOTUMKDM4EIMPDH2ALDH1A1PRMT3
SCHEMBL14456055 0.79 LMNA (0.57) NOTUMIMPDH2
SCHEMBL19860105 0.79 PRMT3 (0.62) NOTUMIMPDH2PRMT3
SCHEMBL19860108 0.79 MEN1 (0.54) NOTUMKDM4EIMPDH2ALDH1A1PRMT3
SCHEMBL3598434 0.78 IMPDH2 (0.69) NOTUMIMPDH2PRMT3ROCK2ROCK1
SCHEMBL19860125 0.78 PRMT3 (0.71) NOTUMIMPDH2PRMT3ROCK2ROCK1
SCHEMBL19860106 0.78 ROCK1 (0.57) NOTUMIMPDH2PRMT3ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed