SCHEMBL19983776

SCHEMBL19983776

CNCc1c[nH]c2cc(-c3cncnc3)ccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.42
CHRNA7 P36544 1/20 0.42
CHRNA4 P43681 1/20 0.42
GPR84 Q9NQS5 2/20 0.39
HASPIN Q8TF76 2/20 0.38
PIM1 P11309 1/20 0.37
PIM3 Q86V86 1/20 0.37
HTR2A P28223 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTR1A P08908 1/20 0.36
HTT P42858 1/20 0.36
SSTR3 P32745 2/20 0.36
IMPDH2 P12268 1/20 0.36
TDO2 P48775 1/20 0.36
ROCK2 O75116 3/20 0.35
ROCK1 Q13464 3/20 0.35
DYRK1A Q13627 1/20 0.35
NR4A2 P43354 1/20 0.35
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19984200 0.82 ROCK2 (0.41) CHRNB2CHRNA7CHRNA4GPR84HTR2A
SCHEMBL19984287 0.77 MAPT (0.45) CHRNB2CHRNA7CHRNA4GPR84HTR2A
SCHEMBL19983953 0.77 GPR84 (0.43) CHRNB2CHRNA7CHRNA4GPR84HTR2A
SCHEMBL19983923 0.77 GPR84 (0.51) CHRNB2CHRNA7CHRNA4GPR84HTR2A
SCHEMBL3281375 0.74 HTR2A (0.61) CHRNB2CHRNA7CHRNA4GPR84HTR2A
SCHEMBL19983810 0.74 ALKBH5 (0.39) CHRNB2CHRNA7CHRNA4GPR84
SCHEMBL31415127 0.73 GPR84 (0.72) CHRNB2CHRNA7CHRNA4GPR84HTR2A
SCHEMBL15897700 0.73 CHRNB2 (0.72) CHRNB2CHRNA7CHRNA4GPR84HTR2A
SCHEMBL25356584 0.72 PTPRA (0.58) PIM1PIM3HTR2AKDM4EALDH1A1
SCHEMBL25356587 0.72 PTPRA (0.58) PIM1PIM3HTR2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed