SCHEMBL19984200

SCHEMBL19984200

CNCc1c[nH]c2cc(-c3cnc(OC)nc3)ccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.41
ROCK1 Q13464 3/20 0.41
TDO2 P48775 2/20 0.40
FTO Q9C0B1 2/20 0.40
PRKACA P17612 1/20 0.39
PRKACG P22612 1/20 0.39
PRKACB P22694 1/20 0.39
HTR2A P28223 2/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA7 P36544 1/20 0.39
CHRNA4 P43681 1/20 0.39
GPR84 Q9NQS5 1/20 0.38
PTGDR Q13258 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
DYRK1B Q9Y463 1/20 0.37
HTR6 P50406 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19983776 0.82 CHRNB2 (0.42) ROCK2ROCK1TDO2HTR2ACHRNB2
SCHEMBL19983953 0.78 GPR84 (0.43) TDO2HTR2ACHRNB2CHRNA7CHRNA4
SCHEMBL19984287 0.76 MAPT (0.45) TDO2HTR2ACHRNB2CHRNA7CHRNA4
SCHEMBL19983923 0.73 GPR84 (0.51) HTR2ACHRNB2CHRNA7CHRNA4GPR84
SCHEMBL31415127 0.72 GPR84 (0.72) TDO2FTOHTR2ACHRNB2CHRNA7
SCHEMBL3281375 0.70 HTR2A (0.61) FTOHTR2ACHRNB2CHRNA7CHRNA4
SCHEMBL19983810 0.70 ALKBH5 (0.39) FTOCHRNB2CHRNA7CHRNA4GPR84
SCHEMBL19983869 0.70 MMP2 (0.46) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL15897700 0.69 CHRNB2 (0.72) HTR2ACHRNB2CHRNA7CHRNA4GPR84
SCHEMBL19983831 0.69 HTR2A (0.49) HTR2AGPR84MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed