SCHEMBL19983810

SCHEMBL19983810

CNCc1c[nH]c2cc(-c3ccnn3C)ccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALKBH5 Q6P6C2 2/20 0.39
FTO Q9C0B1 2/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA7 P36544 1/20 0.39
CHRNA4 P43681 1/20 0.39
HAVCR2 Q8TDQ0 1/20 0.38
ATR Q13535 2/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
LRRK2 Q5S007 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
PI4KA P42356 1/20 0.36
PIK3CG P48736 1/20 0.36
PI4KB Q9UBF8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19983776 0.74 CHRNB2 (0.42) CHRNB2CHRNA7CHRNA4GPR84
SCHEMBL19984287 0.73 MAPT (0.45) CHRNB2CHRNA7CHRNA4CYP3A4CYP2C9
SCHEMBL3281375 0.70 HTR2A (0.61) ALKBH5FTOCHRNB2CHRNA7CHRNA4
SCHEMBL19983923 0.70 GPR84 (0.51) CHRNB2CHRNA7CHRNA4GPR84
SCHEMBL19984200 0.70 ROCK2 (0.41) FTOCHRNB2CHRNA7CHRNA4SMN1; SMN2
SCHEMBL31415127 0.69 GPR84 (0.72) ALKBH5FTOCHRNB2CHRNA7CHRNA4
SCHEMBL15897700 0.69 CHRNB2 (0.72) CHRNB2CHRNA7CHRNA4GPR84
SCHEMBL19983953 0.68 GPR84 (0.43) CHRNB2CHRNA7CHRNA4GPR84
SCHEMBL19984170 0.68 HTR2A (0.44) ALKBH5FTOCHRNB2CHRNA7CHRNA4
SCHEMBL19984283 0.68 HTR2A (0.47) ALKBH5FTOCHRNB2CHRNA7CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed