SCHEMBL19983900

SCHEMBL19983900

CNCc1c[nH]c2cc(Nc3ccc(OC(F)(F)F)cc3C)ccc12

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 1/20 0.42
GOT1 P17174 1/20 0.38
TRPA1 O75762 1/20 0.38
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
P2RX7 Q99572 6/20 0.35
TRPV1 Q8NER1 3/20 0.35
STING1 Q86WV6 1/20 0.35
HTR6 P50406 3/20 0.35
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34
HTR1A P08908 1/20 0.33
HTR7 P34969 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19983859 0.89 CDK2 (0.41) CDK2GOT1TRPA1IDO1TDO2
SCHEMBL19984222 0.88 CDK2 (0.41) CDK2GOT1TRPA1IDO1TDO2
SCHEMBL19984215 0.87 GAA (0.47) CDK2HTR6GAA
SCHEMBL19983847 0.85 TBXAS1 (0.42) CDK2GOT1TRPA1TRPV1HTR1A
SCHEMBL19984134 0.84 HTR2A (0.41) CDK2TRPV1HTR6HTR1A
SCHEMBL19983891 0.82 GPR84 (0.49) HTR6HTR1A
SCHEMBL19984005 0.82 HTR2A (0.44)
SCHEMBL19984189 0.81 BRD4 (0.38) CDK2GOT1TRPV1HTR6HTR1A
SCHEMBL19983867 0.80 HTR2C (0.42) HTR6HTR1AGAA
SCHEMBL19984197 0.80 GPR84 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed