SCHEMBL20003224

SCHEMBL20003224

O=C(C1CCCCC1)N1CC[C@H](Sc2ccc(P)cc2)C1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.43
TSHR P16473 2/20 0.42
ALDH1A1 P00352 1/20 0.42
PTPN1 P18031 1/20 0.40
KEAP1 Q14145 1/20 0.40
HSD11B1 P28845 6/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
HSD11B2 P80365 2/20 0.38
MEN1 O00255 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002719 0.87 HSD11B1 (0.48) KMT2ATSHRALDH1A1PTPN1KEAP1
SCHEMBL20003196 0.87 HSD11B1 (0.48) KMT2ATSHRALDH1A1PTPN1KEAP1
SCHEMBL20003223 0.84 KMT2A (0.41) KMT2ATSHRALDH1A1PTPN1KEAP1
SCHEMBL20003227 0.75 KMT2A (0.38) KMT2ASMN1; SMN2
SCHEMBL20002255 0.74 CCR5 (0.49) KMT2AHSD11B1
SCHEMBL20002972 0.74 L3MBTL1 (0.41) KMT2AHSD11B1
SCHEMBL20003069 0.69 RORC (0.42) KMT2AALDH1A1
SCHEMBL20003024 0.68 NOTUM (0.44) KMT2AALDH1A1HSD11B1MEN1
SCHEMBL20002886 0.67 KMT2A (0.40) KMT2AALDH1A1HSD11B1SMN1; SMN2
SCHEMBL20002297 0.65 NOTUM (0.47) KMT2AHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed