SCHEMBL20002727

SCHEMBL20002727

CCOC(=O)C(Cc1c(F)ccc(F)c1F)C(=O)OCC

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 1/20 0.41
KMT2A Q03164 5/20 0.40
ALDH1A1 P00352 5/20 0.39
TSHR P16473 3/20 0.39
TDP1 Q9NUW8 6/20 0.39
MEN1 O00255 4/20 0.39
KDM4E B2RXH2 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PIN1 Q13526 1/20 0.36
ATM Q13315 1/20 0.35
NPC1 O15118 1/20 0.35
MAPK1 P28482 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
TP53 P04637 1/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5736978 0.85 KMT2A (0.50) MMP8KMT2AALDH1A1TSHRTDP1
SCHEMBL10693803 0.80 MMP8 (0.39) MMP8KMT2AALDH1A1TSHRTDP1
SCHEMBL5737042 0.79 KMT2A (0.48) MMP8KMT2AALDH1A1TSHRTDP1
SCHEMBL3714554 0.78 KMT2A (0.45) MMP8KMT2AALDH1A1TSHRTDP1
SCHEMBL23203481 0.78 ALDH1A1 (0.43) MMP8KMT2AALDH1A1TSHRTDP1
SCHEMBL28297783 0.77 MAPT (0.36) KMT2AALDH1A1TDP1MEN1KDM4E
SCHEMBL7494802 0.76 NLRP3 (0.42) KMT2AALDH1A1TSHRTDP1MEN1
SCHEMBL16342407 0.75 TSHR (0.41) MMP8KMT2AALDH1A1TSHRTDP1
SCHEMBL3412295 0.75 PTGS2 (0.44) KMT2ASMN1; SMN2
SCHEMBL6904885 0.75 CES2 (0.44) MMP8KMT2AALDH1A1TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020246903-A1 DOPAMINE-Β-HYDROXYLASE INHIBITORS BIAL - PORTELA & Cª, S.A. (PT) 2020-12-10 WO disclosed
WO-2018056854-A1 BLOOD-BRAIN BARRIER-PENETRANT DOPAMINE-B-HYDROXYLASE INHIBITORS BIAL - PORTELA & Cª, S.A. (PT) 2018-03-29 WO disclosed
WO-2018056855-A1 DOPAMINE-B-HYDROXYLASE INHIBITORS BIAL - PORTELA & Cª, S.A. (PT) 2018-03-29 WO disclosed