SCHEMBL20002736

SCHEMBL20002736

Cc1cc(S[C@H]2CCN(C(=O)C3(C)CCCCC3)C2)ccc1F

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.36
GRM1 Q13255 1/20 0.36
SLC9A1 P19634 1/20 0.35
HSD11B1 P28845 2/20 0.35
USP19 O94966 2/20 0.35
FASN P49327 3/20 0.35
KMT2A Q03164 2/20 0.34
TACR3 P29371 1/20 0.34
PDE2A O00408 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
GRM2 Q14416 2/20 0.32
GRM3 Q14832 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003055 0.76 RORC (0.42) RORCHSD11B1KMT2ASMN1; SMN2
SCHEMBL20003069 0.76 RORC (0.42) RORCKMT2A
SCHEMBL20002683 0.73 KMT2A (0.39) RORCHSD11B1KMT2A
SCHEMBL20002823 0.70 CCR5 (0.38) HSD11B1KMT2ASMN1; SMN2
SCHEMBL20002294 0.68 PTPN11 (0.36) RORCKMT2A
SCHEMBL20003154 0.67 RORC (0.39) RORCHSD11B1KMT2ASMN1; SMN2
SCHEMBL20002612 0.67 RORC (0.36) RORCKMT2A
SCHEMBL20003220 0.67 RORC (0.41) RORCHSD11B1KMT2ASMN1; SMN2
SCHEMBL29087365 0.66 NPC1 (0.46) SMN1; SMN2
SCHEMBL18703632 0.65 GPR119 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed