SCHEMBL20002683

SCHEMBL20002683

Cc1cc(SC2CCN(C(=O)C3CC[S+]([O-])CC3)C2)ccc1F

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.39
RORC P51449 3/20 0.34
GFER P55789 1/20 0.33
GRIN2B Q13224 4/20 0.33
PIK3CD O00329 1/20 0.33
MTNR1B P49286 1/20 0.33
FPR1 P21462 2/20 0.32
FPR2 P25090 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 2/20 0.32
THRB P10828 1/20 0.32
HSD11B1 P28845 1/20 0.31
GAA P10253 2/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003069 0.86 RORC (0.42) KMT2ARORCGFERGRIN2BPIK3CD
SCHEMBL20002736 0.73 RORC (0.36) KMT2ARORCHSD11B1
SCHEMBL20002255 0.71 CCR5 (0.49) KMT2ARORCHSD11B1
SCHEMBL20003196 0.71 HSD11B1 (0.48) KMT2AALDH1A1HSD11B1
SCHEMBL20002719 0.71 HSD11B1 (0.48) KMT2AALDH1A1HSD11B1
SCHEMBL20002886 0.67 KMT2A (0.40) KMT2ARORCGRIN2BALDH1A1HSD11B1
SCHEMBL20003224 0.66 KMT2A (0.43) KMT2AALDH1A1HSD11B1
SCHEMBL20003152 0.66 RAB9A (0.34) KMT2AGRIN2BALDH1A1MAPTHSD11B1
SCHEMBL20002684 0.65 L3MBTL1 (0.47) RORCALDH1A1MAPTGAAKDM4E
SCHEMBL20002927 0.65 ALDH1A1 (0.46) RORCGFERALDH1A1HSD11B1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed