SCHEMBL20002796

SCHEMBL20002796

CC(C)(O)C12CCC(C(=O)N3CCC([S+]([O-])c4ccc(F)cc4)C3)(CC1)C2

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.45
PDK2 Q15119 6/20 0.32
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
ATM Q13315 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002856 0.86 RORC (0.42) RORCNPC1RAB9AATMALDH1A1
SCHEMBL20003241 0.85 RORC (0.41) RORCNPC1RAB9AATMALDH1A1
SCHEMBL20003044 0.83 RORC (0.40) RORCNPC1RAB9AATMALDH1A1
SCHEMBL20002828 0.78 RORC (0.54) RORC
SCHEMBL20002926 0.78 RORC (0.43) RORC
SCHEMBL20002508 0.78 RORC (0.35) RORCPDK2SMN1; SMN2
SCHEMBL20002171 0.77 KMT2A (0.38) RORCNPC1RAB9AATMSMN1; SMN2
SCHEMBL20002870 0.76 PDK2 (0.38) RORCPDK2ALDH1A1SMN1; SMN2
SCHEMBL20003052 0.75 HSD11B1 (0.38) RORCNPC1RAB9AATMALDH1A1
SCHEMBL20002748 0.75 RORC (0.39) RORCNPC1RAB9AATMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed