SCHEMBL20002956

SCHEMBL20002956

CC(C)(C(=O)N1CCC([S+]([O-])c2ccc(F)cc2)C1)n1cncn1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.44
CYP19A1 P11511 1/20 0.40
MGLL Q99685 8/20 0.35
NTRK1 P04629 1/20 0.35
LMNA P02545 1/20 0.35
FAAH O00519 3/20 0.35
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
PDK2 Q15119 2/20 0.33
GPR119 Q8TDV5 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002210 0.84 RORC (0.44) RORCLMNADRD2DRD4DRD3
SCHEMBL20002870 0.80 PDK2 (0.38) RORCLMNADRD2DRD4DRD3
SCHEMBL20002931 0.78 PDK2 (0.39) RORCDRD2DRD4DRD3PDK2
SCHEMBL20002917 0.77 MEN1 (0.47) GPR119POLB
SCHEMBL20002981 0.74 KDM4E (0.55) LMNAPOLB
SCHEMBL4773698 0.72 MEN1 (0.51) GPR119POLB
SCHEMBL20003082 0.72 SMN1; SMN2 (0.44) RORCCYP19A1LMNAPOLB
SCHEMBL20002167 0.71 KDM1A (0.40) RORCLMNAFAAH
SCHEMBL20002280 0.71 TACR1 (0.40) RORC
SCHEMBL20002631 0.70 HSD11B1 (0.33) RORCLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed