SCHEMBL2000835

SCHEMBL2000835

COc1ccc2c(c1)c(C(=O)c1noc(-c3ccccn3)n1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 5/20 0.38
TP53 P04637 2/20 0.35
MAPT P10636 2/20 0.35
ALOX5AP P20292 1/20 0.35
PTGS2 P35354 1/20 0.35
F2RL3 Q96RI0 3/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C9 P11712 2/20 0.35
ACHE P22303 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
GRM5 P41594 1/20 0.34
GPR39 O43194 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003268 0.94 ALOX5AP (0.36) TP53MAPTALOX5APF2RL3CYP2C9
SCHEMBL2004941 0.93 GRM5 (0.38) TP53MAPTCYP2D6CYP2C9CYP1A2
SCHEMBL2002685 0.91 PLA2G2A (0.37) PLA2G2ATP53MAPTALOX5APPTGS2
SCHEMBL2006492 0.91 GRM5 (0.35) MAPTALOX5APCYP2D6CYP2C9CYP1A2
SCHEMBL2001297 0.90 PLA2G2A (0.38) PLA2G2ATP53MAPTALOX5APACHE
SCHEMBL2002391 0.90 L3MBTL1 (0.39) MAPTALOX5APCYP2D6CYP2C9CYP1A2
SCHEMBL2002093 0.90 LMNA (0.40) TP53MAPTCYP2D6CYP2C9CYP1A2
SCHEMBL4564522 0.89 NPC1 (0.38) PLA2G2ATP53MAPTALOX5APPTGS2
SCHEMBL2003372 0.88 PLA2G2A (0.38) PLA2G2AMAPTALOX5APPTGS2F2RL3
SCHEMBL2001214 0.88 PLA2G2A (0.38) PLA2G2ATP53MAPTPTGS2F2RL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed