SCHEMBL2006492

SCHEMBL2006492

Cc1ccc2c(c1)c(C(=O)c1noc(-c3ccccn3)n1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
CYP2C19 P33261 2/20 0.35
GPR39 O43194 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
LMNA P02545 5/20 0.34
OPRK1 P41145 3/20 0.34
FAAH O00519 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
CES1 P23141 1/20 0.34
GRM4 Q14833 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
TSHR P16473 1/20 0.34
ALOX12 P18054 1/20 0.34
HTT P42858 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004941 0.95 GRM5 (0.38) GRM5MEN1KMT2ANPSR1CYP2C19
SCHEMBL2002391 0.92 L3MBTL1 (0.39) GRM5MEN1KMT2ANPSR1CYP2C19
SCHEMBL2002093 0.92 LMNA (0.40) GRM5MEN1KMT2ANPSR1CYP2C19
SCHEMBL2000835 0.91 PLA2G2A (0.38) GRM5GPR39CYP1A2CYP2D6CYP2C9
SCHEMBL2009499 0.90 FAAH (0.33) MEN1KMT2ANPSR1CYP2C19CYP1A2
SCHEMBL2003537 0.90 GRM5 (0.38) GRM5MEN1KMT2ANPSR1CYP2C19
SCHEMBL2003268 0.90 ALOX5AP (0.36) GRM5GPR39CYP2C9LMNAFAAH
SCHEMBL2009569 0.87 GRM5 (0.39) GRM5MEN1KMT2ANPSR1CYP2C19
SCHEMBL2008461 0.87 RET (0.36) MEN1KMT2ACYP2C9LMNAFAAH
SCHEMBL1999092 0.87 L3MBTL1 (0.42) GRM5MEN1KMT2ANPSR1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed