SCHEMBL20008765

SCHEMBL20008765

C=CCCN(CCC)c1cc(-c2cccnc2C)cc(N2CCCCC2)n1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1B Q01064 4/20 0.33
KDM4E B2RXH2 5/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
USP2 O75604 1/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
CNR2 P34972 1/20 0.33
PDE1A P54750 3/20 0.33
NMT1 P30419 3/20 0.32
PDE1C Q14123 2/20 0.32
CRHR1 P34998 3/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PTPN11 Q06124 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20008457 0.83 L3MBTL1 (0.34) KDM4EALDH1A1HPGDHSD17B10TDP1
SCHEMBL20010275 0.71
SCHEMBL20008830 0.70 RAF1 (0.34) CRHR1
SCHEMBL20009409 0.69 RAF1 (0.45) KDM4EALDH1A1HPGDHSD17B10TDP1
SCHEMBL20008434 0.68 CRHR1 (0.34) CRHR1
SCHEMBL7718046 0.64 SMN1; SMN2 (0.43) KDM4EALDH1A1LMNATSHRCRHR1
SCHEMBL15730626 0.63 CNR2 (0.64) KDM4ECNR2
SCHEMBL25925332 0.60 AGTR1 (0.36) CRHR1L3MBTL1KMT2A
SCHEMBL23916149 0.60 S1PR1 (0.32) CRHR1
SCHEMBL20008328 0.59 CNR2 (0.48) KDM4EALDH1A1HPGDHSD17B10TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed