SCHEMBL20009430

SCHEMBL20009430

Cc1ccc(C)c(-c2cc(-c3c(C)n[nH]c3C)nc(N3CCCC3)c2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 2/20 0.49
BRAF P15056 1/20 0.49
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
AR P10275 1/20 0.37
ATR Q13535 3/20 0.36
KMT2A Q03164 1/20 0.36
LRRK2 Q5S007 2/20 0.35
ATRIP Q8WXE1 1/20 0.34
KDM4E B2RXH2 3/20 0.34
GAA P10253 3/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
MAPK1 P28482 1/20 0.34
ATM Q13315 1/20 0.34
CLK2 P49760 2/20 0.34
CLK3 P49761 2/20 0.34
DYRK1A Q13627 2/20 0.34
BRD4 O60885 1/20 0.34
KCNH2 Q12809 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20008452 0.74 GALR2 (0.44) KMT2AKDM4EGAAL3MBTL1MAPK1
SCHEMBL20008122 0.73 SMN1; SMN2 (0.46) RAF1BRAFKMT2AKDM4EGAA
SCHEMBL20008237 0.71 HRH4 (0.47) RAF1BRAFLRRK2
SCHEMBL20008538 0.70 DRD2 (0.49) RAF1ARKMT2AKDM4EGAA
SCHEMBL20008460 0.70 RAF1 (0.41) RAF1BRAFARKMT2AKDM4E
SCHEMBL20009412 0.70 RAF1 (0.40) RAF1BRAFARKMT2AKDM4E
SCHEMBL19529392 0.70 RAF1 (0.40) RAF1BRAFARKMT2AKDM4E
SCHEMBL20010376 0.65 AR (0.53) RAF1BRAFARATRKMT2A
SCHEMBL2166402 0.65 HRH4 (0.55) HRH3
SCHEMBL13575902 0.63 ALDH1A1 (0.43) ATRKMT2AATRIPKDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed