SCHEMBL20022707

SCHEMBL20022707

O=c1c2ccccc2sn1CN1CCN(Cc2ccccc2)CC1

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 6/20 0.68
P4HB P07237 1/20 0.60
FAAH O00519 1/20 0.58
MGLL Q99685 1/20 0.58
SIGMAR1 Q99720 1/20 0.50
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
KAT2A Q92830 1/20 0.47
KAT2B Q92831 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17948281 0.90 P4HB (0.71) CASP3P4HBFAAHMGLL
SCHEMBL11640205 0.88 CASP3 (0.67) CASP3FAAHMGLLKAT2AKAT2B
SCHEMBL17948336 0.83 P4HB (0.63) CASP3P4HBFAAHMGLLKAT2A
SCHEMBL17948283 0.83 P4HB (0.63) CASP3P4HBFAAHMGLL
SCHEMBL24766317 0.82 P4HB (0.62) CASP3P4HBFAAHMGLL
SCHEMBL17948289 0.82 P4HB (0.62) CASP3P4HBFAAHMGLL
SCHEMBL79203 0.82 CASP3 (1.00) CASP3FAAHMGLLHDAC3HDAC4
SCHEMBL17948284 0.81 P4HB (0.61) CASP3P4HBFAAHMGLLKAT2A
SCHEMBL22056074 0.81 KAT2B (0.72) CASP3SIGMAR1HDAC3HDAC1HDAC8
SCHEMBL10833057 0.80 P4HB (0.60) CASP3P4HB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240216365-A1 METHODS AND USES OF PROTEIN DISULFIDE ISOMERASE INHIBITORY COMPOUNDS THE UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2024-07-04 US disclosed
US-20240216365-A1 METHODS AND USES OF PROTEIN DISULFIDE ISOMERASE INHIBITORY COMPOUNDS THE UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2024-07-04 US disclosed
US-20210353620-A1 METHODS AND USES OF PROTEIN DISULFIDE ISOMERASE INHIBITORY COMPOUNDS THE UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE 2021-11-18 US disclosed
US-20180092908-A1 SMALL MOLECULE OXIDIZERS OF PDI AND THEIR USE THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2018-04-05 US disclosed
US-20180092908-A1 SMALL MOLECULE OXIDIZERS OF PDI AND THEIR USE THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2018-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210353620-A1 METHODS AND USES OF PROTEIN DISULFIDE ISOMERASE INHIBITORY COMPOUNDS PDIA3, PDIA4, PDIA5 CASP3 1339/4885P4HB 5/4885FAAH 1576/4885
US-20180092908-A1 SMALL MOLECULE OXIDIZERS OF PDI AND THEIR USE PDIA5, PDIA4, PDIA6 CASP3 2233/4885P4HB 5/4885FAAH 2785/4885
US-20240216365-A1 METHODS AND USES OF PROTEIN DISULFIDE ISOMERASE INHIBITORY COMPOUNDS PDIA3, PDIA4, PDIA5 CASP3 1339/4885P4HB 5/4885FAAH 1576/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.