SCHEMBL20042690

SCHEMBL20042690

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)CCc1ccncc1)C2

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GFER P55789 2/20 0.41
CHRM4 P08173 2/20 0.40
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
LMNA P02545 1/20 0.39
GPBAR1 Q8TDU6 3/20 0.37
NPC1 O15118 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
GRM5 P41594 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
NAAA Q02083 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042748 0.90 NPC1 (0.49) GFERALDH1A1MEN1KMT2AGPBAR1
SCHEMBL20042830 0.88 ME2 (0.43) ALDH1A1MEN1KMT2AGPBAR1NPC1
SCHEMBL20042688 0.88 C3AR1 (0.45) CHRM4MEN1KMT2A
SCHEMBL20042747 0.84 GRIN1 (0.39) KMT2AGPBAR1
SCHEMBL20042703 0.83 PTGDR2 (0.37) CHRM4
SCHEMBL20042673 0.81 MAPK1 (0.38)
SCHEMBL20042714 0.78 CHRM4 (0.43) CHRM4ALDH1A1KMT2ALMNA
SCHEMBL20042654 0.77 HSD11B1 (0.41) CHRM4ALDH1A1MEN1KMT2ALMNA
SCHEMBL20042834 0.75 CHRM4 (0.56) CHRM4ALDH1A1LMNA
SCHEMBL20042651 0.74 CHRM4 (0.52) CHRM4ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed