SCHEMBL2006172

SCHEMBL2006172

CCOc1ccc2c(c1)c(C(=O)c1cnc(-c3cccnc3)o1)c(Cl)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 5/20 0.39
ALOX5 P09917 2/20 0.39
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
LMNA P02545 3/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
MAPT P10636 3/20 0.36
RXFP1 Q9HBX9 2/20 0.36
P2RX7 Q99572 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NTRK1 P04629 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
SLC26A4 O43511 1/20 0.35
POLB P06746 1/20 0.35
PTGES2 Q9H7Z7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003889 0.93 ALDH1A1 (0.38) ALOX5APALOX5CYP3A4CYP2C9LMNA
SCHEMBL2011328 0.92 LMNA (0.40) ALOX5APCYP3A4CYP2D6CYP2C9LMNA
SCHEMBL2002164 0.92 ALOX5AP (0.45) ALOX5APALOX5CYP3A4CYP2D6CYP2C9
SCHEMBL2007346 0.92 ALOX5AP (0.39) ALOX5APALOX5CYP3A4CYP2D6CYP2C9
SCHEMBL2003941 0.91 P2RX7 (0.38) CYP3A4CYP2D6CYP2C9LMNAHTT
SCHEMBL2008130 0.91 ALOX5AP (0.39) ALOX5APALOX5CYP3A4CYP2D6CYP2C9
SCHEMBL1996791 0.89 PTGES2 (0.38) ALOX5APCYP3A4CYP2D6CYP2C9LMNA
SCHEMBL2006961 0.89 LMNA (0.40) ALOX5APALOX5CYP3A4LMNAMAPK1
SCHEMBL2002287 0.88 L3MBTL1 (0.39) ALOX5APALOX5CYP3A4CYP2D6CYP2C9
SCHEMBL2008737 0.88 LMNA (0.42) CYP3A4CYP2D6CYP2C9LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed