SCHEMBL20042688

SCHEMBL20042688

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)CCc1cccnc1)C2

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
C3AR1 Q16581 12/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.42
RAB9A P51151 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CHRM4 P08173 2/20 0.42
CYP1A2 P05177 1/20 0.42
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042748 0.89 NPC1 (0.49) MEN1KMT2APOLB
SCHEMBL20042690 0.88 GFER (0.41) MEN1KMT2ACHRM4
SCHEMBL20042750 0.83 F2 (0.39) MEN1KMT2A
SCHEMBL20042830 0.83 ME2 (0.43) MEN1KMT2A
SCHEMBL20042832 0.81 CFTR (0.45) MEN1KMT2AKDM4EPOLB
SCHEMBL20042747 0.80 GRIN1 (0.39) PTGDR2KMT2A
SCHEMBL20042888 0.80 PTGDR2 (0.35) PTGDR2CHRM4CYP1A2
SCHEMBL20042703 0.80 PTGDR2 (0.37) PTGDR2CHRM4CYP1A2
SCHEMBL20042673 0.78 MAPK1 (0.38) PTGDR2
SCHEMBL20042714 0.75 CHRM4 (0.43) KMT2ACHRM4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed