SCHEMBL20042703

SCHEMBL20042703

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)CCc1ccc(F)c(C)c1)C2

nearest known ligand 0.37

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 14/20 0.37
CYP1A2 P05177 1/20 0.35
CHRM4 P08173 1/20 0.35
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042888 0.92 PTGDR2 (0.35) PTGDR2CYP1A2CHRM4
SCHEMBL20042673 0.91 MAPK1 (0.38) PTGDR2
SCHEMBL20042830 0.86 ME2 (0.43)
SCHEMBL20042747 0.85 GRIN1 (0.39) PTGDR2GRIN2B
SCHEMBL20042750 0.85 F2 (0.39)
SCHEMBL20042748 0.84 NPC1 (0.49)
SCHEMBL20042690 0.83 GFER (0.41) CHRM4
SCHEMBL20042836 0.81 P2RX7 (0.43)
SCHEMBL20042688 0.80 C3AR1 (0.45) PTGDR2CYP1A2CHRM4
SCHEMBL20042666 0.76 KMT2A (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed