SCHEMBL20042747

SCHEMBL20042747

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)CCc1ccc(Cl)c(Cl)c1)C2

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.37
CXCR3 P49682 1/20 0.37
P2RY12 Q9H244 1/20 0.36
KMT2A Q03164 1/20 0.36
AIMP2 Q13155 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
KCNQ2 O43526 1/20 0.35
SMYD2 Q9NRG4 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35
OPRK1 P41145 1/20 0.35
CCR2 P41597 1/20 0.34
FKBP1A P62942 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042673 0.92 MAPK1 (0.38) PTGDR2AIMP2
SCHEMBL20042830 0.89 ME2 (0.43) KMT2AGPBAR1FKBP1A
SCHEMBL20042750 0.87 F2 (0.39) KMT2AKCNQ2
SCHEMBL20042888 0.85 PTGDR2 (0.35) PTGDR2GPBAR1
SCHEMBL20042703 0.85 PTGDR2 (0.37) GRIN2BPTGDR2
SCHEMBL20042748 0.85 NPC1 (0.49) KMT2AGPBAR1FKBP1A
SCHEMBL20042690 0.84 GFER (0.41) KMT2AGPBAR1
SCHEMBL20042886 0.81 HPGD (0.49) KMT2A
SCHEMBL20042688 0.80 C3AR1 (0.45) PTGDR2KMT2A
SCHEMBL20042887 0.76 GPR6 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed