SCHEMBL20042832

SCHEMBL20042832

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1cccnc1)C2

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.45
HPGD P15428 1/20 0.45
MAPK1 P28482 1/20 0.45
P2RX7 Q99572 1/20 0.43
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 2/20 0.43
FABP6 P51161 1/20 0.43
GAA P10253 1/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PKM P14618 1/20 0.42
POLB P06746 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042776 0.88 P2RX7 (0.41) CFTRP2RX7MEN1KMT2AKDM4E
SCHEMBL20042839 0.88 P2RX7 (0.45) CFTRHPGDP2RX7MEN1MAPT
SCHEMBL20042755 0.86 GRM5 (0.43) HPGDP2RX7MEN1KMT2AALDH1A1
SCHEMBL20042873 0.86 P2RX7 (0.38) CFTRHPGDP2RX7MEN1KMT2A
SCHEMBL20042674 0.84 P2RX7 (0.37) CFTRP2RX7MEN1KMT2ATDP1
SCHEMBL20042668 0.83 HPGD (0.51) HPGDP2RX7MEN1KMT2AALDH1A1
SCHEMBL20042817 0.83 PKM (0.44) HPGDP2RX7MEN1KMT2AALDH1A1
SCHEMBL20042771 0.82 P2RX7 (0.47) HPGDP2RX7MEN1MAPTKMT2A
SCHEMBL20042684 0.82 SMN1; SMN2 (0.52) HPGDMAPK1P2RX7TDP1ALDH1A1
SCHEMBL20042872 0.81 P2RX7 (0.44) CFTRP2RX7SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed