SCHEMBL20042888

SCHEMBL20042888

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)CCc1ccc(C)c(F)c1)C2

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 10/20 0.35
CHRM4 P08173 2/20 0.35
CYP1A2 P05177 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35
P2RX7 Q99572 1/20 0.35
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042703 0.92 PTGDR2 (0.37) PTGDR2CHRM4CYP1A2
SCHEMBL20042673 0.89 MAPK1 (0.38) PTGDR2P2RX7
SCHEMBL20042747 0.85 GRIN1 (0.39) PTGDR2GPBAR1
SCHEMBL20042830 0.84 ME2 (0.43) GPBAR1MAPT
SCHEMBL20042748 0.84 NPC1 (0.49) GPBAR1MAPT
SCHEMBL20042690 0.83 GFER (0.41) CHRM4GPBAR1
SCHEMBL20042750 0.83 F2 (0.39) MAPT
SCHEMBL20042823 0.81 P2RX7 (0.45) P2RX7
SCHEMBL20042688 0.80 C3AR1 (0.45) PTGDR2CHRM4CYP1A2
SCHEMBL20042836 0.75 P2RX7 (0.43) P2RX7MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed