SCHEMBL20042873

SCHEMBL20042873

Cc1cncc(C(=O)N2Cc3nc(C)nc(N4CCC4)c3C2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.38
HCAR2 Q8TDS4 1/20 0.37
CFTR P13569 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HPGD P15428 2/20 0.35
ATM Q13315 1/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
HSP90AA1 P07900 3/20 0.34
GBA1 P04062 3/20 0.33
KDM4E B2RXH2 2/20 0.33
TSHR P16473 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
PIK3C3 Q8NEB9 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.33
HSP90B1 P14625 1/20 0.33
IDH1 O75874 1/20 0.33
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042674 0.89 P2RX7 (0.37) P2RX7HCAR2CFTRMEN1KMT2A
SCHEMBL20042832 0.86 CFTR (0.45) P2RX7CFTRMEN1KMT2AHPGD
SCHEMBL20042668 0.84 HPGD (0.51) P2RX7MEN1KMT2AHPGDGBA1
SCHEMBL20042776 0.84 P2RX7 (0.41) P2RX7HCAR2CFTRMEN1KMT2A
SCHEMBL20042817 0.84 PKM (0.44) P2RX7MEN1KMT2AHPGDGBA1
SCHEMBL20042743 0.84 P2RX7 (0.40) P2RX7HPGDGBA1KDM4ETSHR
SCHEMBL20042854 0.83 GRM5 (0.42) P2RX7MEN1KMT2AHPGDHSP90AA1
SCHEMBL20042756 0.83 P2RX7 (0.38) P2RX7MEN1KMT2AHSP90AA1GBA1
SCHEMBL20042755 0.82 GRM5 (0.43) P2RX7MEN1KMT2AHPGDGBA1
SCHEMBL20042689 0.82 P2RX7 (0.39) P2RX7HSP90AA1GBA1CNR2CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed