SCHEMBL20042780

SCHEMBL20042780

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccc(OC(F)(F)F)c(F)c1)C2

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.43
MAPK7 Q13164 1/20 0.36
MGLL Q99685 2/20 0.36
EPHX2 P34913 5/20 0.36
PRLHR P49683 2/20 0.35
GPR6 P46095 2/20 0.35
SLC6A4 P31645 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
GBA1 P04062 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042694 0.93 P2RX7 (0.43) P2RX7MAPK7MGLLPRLHRGPR6
SCHEMBL20042765 0.90 P2RX7 (0.42) P2RX7MAPK7MGLLEPHX2GPR6
SCHEMBL20042917 0.87 P2RX7 (0.39) P2RX7GPR6
SCHEMBL20042666 0.86 KMT2A (0.46) P2RX7GBA1
SCHEMBL20042705 0.85 EPHX2 (0.45) P2RX7MAPK7MGLLEPHX2PRLHR
SCHEMBL20042823 0.85 P2RX7 (0.45) P2RX7PRLHRGBA1
SCHEMBL20042792 0.84 TACR3 (0.46) P2RX7GPR6
SCHEMBL20042836 0.83 P2RX7 (0.43) P2RX7GBA1
SCHEMBL20042882 0.82 P2RX7 (0.41) P2RX7GPR6GBA1
SCHEMBL20042696 0.82 KDM1A (0.45) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed