SCHEMBL20042705

SCHEMBL20042705

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccc(OC(F)(F)F)cc1)C2

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.45
MAPK7 Q13164 5/20 0.44
HRH3 Q9Y5N1 2/20 0.44
P2RX7 Q99572 1/20 0.42
MGLL Q99685 2/20 0.41
HSD11B1 P28845 1/20 0.41
PRLHR P49683 2/20 0.41
LSS P48449 1/20 0.40
TRPM8 Q7Z2W7 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4D Q08499 1/20 0.40
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042707 0.87 P2RX7 (0.40) EPHX2MAPK7P2RX7MGLLTRPM8
SCHEMBL20042704 0.86 P2RX7 (0.50) EPHX2P2RX7
SCHEMBL20042796 0.86 P2RX7 (0.38) P2RX7LMNATP53
SCHEMBL20042694 0.85 P2RX7 (0.43) MAPK7P2RX7MGLLPRLHR
SCHEMBL20042780 0.85 P2RX7 (0.43) EPHX2MAPK7HRH3P2RX7MGLL
SCHEMBL20042861 0.85 P2RX7 (0.39) MAPK7P2RX7MGLL
SCHEMBL20042685 0.85 HTT (0.42) EPHX2P2RX7HSD11B1
SCHEMBL20042817 0.85 PKM (0.44) P2RX7LMNA
SCHEMBL20042765 0.85 P2RX7 (0.42) EPHX2MAPK7P2RX7MGLL
SCHEMBL20042751 0.83 HSD17B10 (0.49) P2RX7MGLLLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed