SCHEMBL20043089

SCHEMBL20043089

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccnc(C(F)(F)F)c1)C2

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.52
CHRM2 P08172 1/20 0.44
CHRM4 P08173 1/20 0.44
PKM P14618 1/20 0.43
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GRM2 Q14416 5/20 0.38
ABL1 P00519 1/20 0.38
BCR P11274 1/20 0.38
PDE4B Q07343 1/20 0.38
BRAF P15056 4/20 0.38
RAF1 P04049 2/20 0.38
SLC6A7 Q99884 1/20 0.37
PROKR1 Q8TCW9 1/20 0.37
SPR P35270 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042872 0.87 P2RX7 (0.44) P2RX7CHRM4LMNASMN1; SMN2HSD17B10
SCHEMBL20042652 0.87 P2RX7 (0.66) P2RX7LMNASMN1; SMN2ABL1BCR
SCHEMBL20042760 0.87 P2RX7 (0.45) P2RX7PKMABL1BCR
SCHEMBL20042704 0.84 P2RX7 (0.50) P2RX7SMN1; SMN2ABL1BCRSLC6A7
SCHEMBL20042697 0.84 PROKR1 (0.48) P2RX7CHRM2CHRM4LMNASMN1; SMN2
SCHEMBL20042701 0.84 PROKR1 (0.47) P2RX7CHRM4LMNASMN1; SMN2HSD17B10
SCHEMBL20042666 0.82 KMT2A (0.46) P2RX7
SCHEMBL20042702 0.82 P2RX7 (0.49) P2RX7SMN1; SMN2HSD17B10
SCHEMBL20042671 0.82 P2RX7 (0.45) P2RX7SMN1; SMN2
SCHEMBL31614786 0.82 CHRM4 (0.52) P2RX7CHRM2CHRM4GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed