SCHEMBL20042760

SCHEMBL20042760

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccc(C(F)(F)F)nc1)C2

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.45
HTR1A P08908 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
PKM P14618 1/20 0.38
KCNH2 Q12809 4/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
CNR2 P34972 1/20 0.37
GBA1 P04062 3/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
ABL1 P00519 1/20 0.36
BCR P11274 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20043089 0.87 P2RX7 (0.52) P2RX7PKMABL1BCR
SCHEMBL20042755 0.86 GRM5 (0.43) P2RX7GBA1MEN1KMT2AABL1
SCHEMBL20042704 0.85 P2RX7 (0.50) P2RX7KCNH2CNR2GBA1MEN1
SCHEMBL20042652 0.82 P2RX7 (0.66) P2RX7MEN1KMT2AABL1BCR
SCHEMBL20042776 0.82 P2RX7 (0.41) P2RX7CNR2GBA1MEN1KMT2A
SCHEMBL20042685 0.82 HTT (0.42) P2RX7KCNH2GBA1CYP1A2CYP2C9
SCHEMBL20042817 0.82 PKM (0.44) P2RX7PKMGBA1MEN1KMT2A
SCHEMBL20042705 0.81 EPHX2 (0.45) P2RX7HRH3
SCHEMBL20042751 0.80 HSD17B10 (0.49) P2RX7KCNH2GBA1MEN1KMT2A
SCHEMBL20042769 0.80 P2RX7 (0.38) P2RX7CNR2GBA1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed