SCHEMBL20042704

SCHEMBL20042704

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccc(C(F)(F)F)cc1)C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.50
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
GBA1 P04062 3/20 0.45
ABL1 P00519 1/20 0.44
BCR P11274 1/20 0.44
KDM1A O60341 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
EPHX2 P34913 3/20 0.42
CNR1 P21554 2/20 0.42
CNR2 P34972 2/20 0.42
SLC6A7 Q99884 1/20 0.42
PHGDH O43175 1/20 0.41
NPY5R Q15761 1/20 0.41
GAA P10253 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042685 0.88 HTT (0.42) P2RX7GBA1ABL1BCRCYP1A2
SCHEMBL20042652 0.88 P2RX7 (0.66) P2RX7MEN1KMT2AHPGDABL1
SCHEMBL20042817 0.88 PKM (0.44) P2RX7MEN1KMT2AHPGDGBA1
SCHEMBL20042705 0.86 EPHX2 (0.45) P2RX7EPHX2
SCHEMBL20042760 0.85 P2RX7 (0.45) P2RX7MEN1KMT2AGBA1ABL1
SCHEMBL20042751 0.85 HSD17B10 (0.49) P2RX7MEN1KMT2AHPGDGBA1
SCHEMBL20042839 0.85 P2RX7 (0.45) P2RX7MEN1KMT2AHPGDTSHR
SCHEMBL20042702 0.85 P2RX7 (0.49) P2RX7MEN1KMT2ATSHRCYP1A2
SCHEMBL20043089 0.84 P2RX7 (0.52) P2RX7ABL1BCRSLC6A7SMN1; SMN2
SCHEMBL20042728 0.83 MEN1 (0.42) MEN1KMT2AGBA1EPHX2SLC6A7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed