SCHEMBL20135538

SCHEMBL20135538

Cc1cc(C(=O)N2CCN(c3ncc(C4CC4)cc3C)CC2)ccc1C1(C(C)C)NC(=O)NC1=O

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 8/20 0.35
ADAM17 P78536 5/20 0.35
FASN P49327 5/20 0.34
MMP2 P08253 2/20 0.34
ADAMTS4 O75173 1/20 0.34
MMP1 P03956 1/20 0.34
MMP12 P39900 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 1/20 0.34
CRBN Q96SW2 1/20 0.34
GPR6 P46095 1/20 0.34
SLC6A7 Q99884 1/20 0.33
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29688547 1.00 ADAMTS5 (0.35) ADAMTS5ADAM17FASNMMP2ADAMTS4
SCHEMBL29688861 0.91 LMNA (0.41) ADAMTS5ADAM17FASNALDH1A1
SCHEMBL20135085 0.91 LMNA (0.41) ADAMTS5ADAM17FASNALDH1A1
SCHEMBL20134769 0.90 SLC6A7 (0.36) ADAMTS5ADAM17FASNMMP2ALDH1A1
SCHEMBL29688685 0.89 ALDH1A1 (0.37) ADAMTS5ADAM17ALDH1A1TSHRCRBN
SCHEMBL20135552 0.89 ALDH1A1 (0.37) ADAMTS5ADAM17ALDH1A1TSHRCRBN
SCHEMBL29688589 0.89 ALDH1A1 (0.37) ADAMTS5ADAM17ALDH1A1TSHRCRBN
SCHEMBL29688455 0.89 ALDH1A1 (0.37) ADAMTS5ADAM17ALDH1A1TSHRCRBN
SCHEMBL20134750 0.89 ALDH1A1 (0.37) ADAMTS5ADAM17ALDH1A1TSHRCRBN
SCHEMBL20134751 0.89 ALDH1A1 (0.37) ADAMTS5ADAM17ALDH1A1TSHRCRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10407408-B2 Imide derivatives and use thereof as medicine MITSUBISHI TANABE PHARMA CORPORATION (JP) 2019-09-10 US disclosed
US-10407408-B2 Imide derivatives and use thereof as medicine MITSUBISHI TANABE PHARMA CORPORATION (JP) 2019-09-10 US disclosed
US-20190077787-A1 NOVEL IMIDE DERIVATIVES AND USE THEREOF AS MEDICINE MITSUBISHI TANABE PHARMA CORPORATION (JP) 2019-03-14 US disclosed
US-20190077787-A1 NOVEL IMIDE DERIVATIVES AND USE THEREOF AS MEDICINE MITSUBISHI TANABE PHARMA CORPORATION (JP) 2019-03-14 US disclosed
EP-3321256-A1 NOVEL IMIDE DERIVATIVES AND USE THEREOF AS MEDICINE Mitsubishi Tanabe Pharma Corporation (JP) 2018-05-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190077787-A1 NOVEL IMIDE DERIVATIVES AND USE THEREOF AS MEDICINE MMP9, MMP10, MMP1 ADAMTS5 23/4885ADAM17 36/4885FASN 4035/4885
US-10407408-B2 Imide derivatives and use thereof as medicine MMP9, MMP2, MMP1 ADAMTS5 25/4885ADAM17 39/4885FASN 4048/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.