SCHEMBL20145073

SCHEMBL20145073

CN1CCC[C@@H](Oc2ncc(C(F)(F)F)cn2)C1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IL1B P01584 1/20 0.50
NLRP3 Q96P20 1/20 0.50
HCRTR1 O43613 8/20 0.41
HCRTR2 O43614 2/20 0.40
CHRM2 P08172 2/20 0.40
CHRM1 P11229 2/20 0.40
CHRM3 P20309 2/20 0.40
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
MAP3K12 Q12852 1/20 0.39
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20144818 1.00 IL1B (0.50) IL1BNLRP3HCRTR1HCRTR2CHRM2
SCHEMBL20144750 0.83 IL1B (0.55) IL1BNLRP3HCRTR1
SCHEMBL20145221 0.83 IL1B (0.55) IL1BNLRP3HCRTR1
SCHEMBL20145042 0.81 PDE3B (0.47) CHRM2CHRM1CHRM3CHRM4CHRM5
SCHEMBL20145182 0.81 IL1B (0.46) IL1BNLRP3HCRTR1
SCHEMBL20145104 0.80 KMT2A (0.46) IL1BNLRP3HCRTR1HCRTR2
SCHEMBL20145101 0.76 IL1B (0.46) IL1BNLRP3HCRTR1CHRM2CHRM1
SCHEMBL20144981 0.76 IL1B (0.46) IL1BNLRP3HCRTR1CHRM2CHRM1
SCHEMBL25072354 0.75 HMOX1 (0.46) HCRTR1HCRTR2
SCHEMBL20145199 0.75 LIPE (0.55) IL1BNLRP3HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed