SCHEMBL20161118

SCHEMBL20161118

N=C(c1nc(N2CCOCC2)n[nH]1)c1cccnc1NCc1ccccc1F

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 4/20 0.46
STAT6 P42226 2/20 0.44
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPT P10636 1/20 0.44
ACHE P22303 2/20 0.41
ABCB1 P08183 1/20 0.41
GAA P10253 1/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PDE5A O76074 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
CDK5 Q00535 1/20 0.37
HTT P42858 1/20 0.36
CSNK1E P49674 2/20 0.36
PTK2 Q05397 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20161209 0.80 AURKA (0.40) KDM4EALDH1A1MAPTGAAPOLB
SCHEMBL20161096 0.80 STAT6 (0.47) CSNK1DSTAT6KDM4EALDH1A1MAPT
SCHEMBL20149081 0.79 KDM4E (0.38) KDM4EGAAPOLBSMN1; SMN2PDE5A
SCHEMBL20161291 0.78 LMNA (0.39) KDM4EALDH1A1GAAPOLBSMN1; SMN2
SCHEMBL20161113 0.77 RPS6KB1 (0.41) KDM4EALDH1A1MAPTGAACCNE1
SCHEMBL20161335 0.76 KDM4E (0.37) STAT6KDM4EALDH1A1MAPTGAA
SCHEMBL20161518 0.75 CASP6 (0.43) KDM4EALDH1A1SMN1; SMN2CCNE1CDK2
SCHEMBL20161340 0.75 CYP11B1 (0.35) KDM4EMAPTMAPK1POLBSMN1; SMN2
SCHEMBL20161268 0.75 ACHE (0.36) KDM4EALDH1A1ACHE
SCHEMBL20161301 0.74 SMN1; SMN2 (0.55) SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089330-A2 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed