SCHEMBL20170612

SCHEMBL20170612

COc1ccc2c3c1OC1C(N)CCC(CC2)C31

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 6/20 0.35
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
HTR1A P08908 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170605 1.00 ADRA1A (0.35) ADRA1ADRD2DRD3HTR1A
SCHEMBL20170607 0.85 OPRM1 (0.37)
SCHEMBL20170652 0.85 OPRM1 (0.37)
SCHEMBL20170728 0.85 OPRM1 (0.37)
SCHEMBL20170740 0.80
SCHEMBL20170753 0.80 GABRA1 (0.39) DRD2
SCHEMBL20170592 0.78 MTNR1A (0.40)
SCHEMBL20170738 0.77 HTR1A (0.40) DRD2DRD3HTR1A
SCHEMBL20170641 0.76 ADRA1A (0.34) ADRA1AHTR1A
SCHEMBL20170640 0.75 HTR1A (0.34) DRD2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed