Benzimidazole

Benzimidazole

SCHEMBL2020186

O=C(O)C(F)(F)F.c1ccc2[nH]cnc2c1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
HTT P42858 2/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HPGD P15428 1/20 0.50
CTNNB1 P35222 2/20 0.47
WNT3A P56704 2/20 0.47
NAMPT P43490 1/20 0.43
POLB P06746 3/20 0.41
MAPT P10636 1/20 0.41
NPC1 O15118 2/20 0.41
PARP1 P09874 2/20 0.41
PDPK1 O15530 1/20 0.41
CA12 O43570 1/20 0.41
ALOX15 P16050 1/20 0.41
CA9 Q16790 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
QPCT Q16769 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzimidazole SCHEMBL29397040 1.00 RAB9A (0.50) RAB9ASMN1; SMN2HTTKDM4EALDH1A1
Benzimidazole SCHEMBL2073386 1.00 RAB9A (0.50) RAB9ASMN1; SMN2HTTKDM4EALDH1A1
Benzimidazole SCHEMBL2075174 1.00 RAB9A (0.50) RAB9ASMN1; SMN2HTTKDM4EALDH1A1
Benzimidazole SCHEMBL28329484 0.94 SMN1; SMN2 (0.46) RAB9ASMN1; SMN2HTTKDM4EALDH1A1
Benzimidazole SCHEMBL16516335 0.87 SMN1; SMN2 (0.57) RAB9ASMN1; SMN2HTTKDM4EALDH1A1
Benzimidazole SCHEMBL8901469 0.87 SMN1; SMN2 (0.57) RAB9ASMN1; SMN2HTTKDM4EALDH1A1
Benzimidazole SCHEMBL4774682 0.85 KDM4E (0.56) RAB9ASMN1; SMN2HTTKDM4EALDH1A1
Benzimidazole SCHEMBL16516333 0.84 KDM4E (0.54) RAB9ASMN1; SMN2HTTKDM4EALDH1A1
Benzimidazole SCHEMBL4631509 0.84 SMN1; SMN2 (0.54) RAB9ASMN1; SMN2HTTKDM4EALDH1A1
Benzimidazole SCHEMBL158526 0.84 SMN1; SMN2 (0.54) RAB9ASMN1; SMN2HTTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581217-A4 CARBONYLAMINO-BENZIMIDAZOLE DERIVATIVES AS ANDROGEN RECEPTOR MODULATORS MERCK & CO INC (US) 2007-07-11 EP claimed
EP-1581217-A1 CARBONYLAMINO-BENZIMIDAZOLE DERIVATIVES AS ANDROGEN RECEPTOR MODULATORS Merck & Co., Inc. (US) 2005-10-05 EP claimed
WO-2004041277-A1 CARBONYLAMINO-BENZIMIDAZOLE DERIVATIVES AS ANDROGEN RECEPTOR MODULATORS MERCK & CO., INC. (US) 2004-05-21 WO claimed
EP-4731306-A1 CYSTOBACTAMID DERIVATIVES Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2026-04-29 EP disclosed
WO-2025003147-A1 CYSTOBACTAMID DERIVATIVES Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2025-01-02 WO disclosed
CN-117986511-A Quaternary ammonium type covalent organic framework compound and preparation method of anion exchange membrane thereof 大连理工大学 2024-05-07 CN disclosed
WO-2021162070-A1 METHOD FOR PRODUCING MONOMER FOR NUCLEIC ACID PRODUCTION 東レ株式会社 2021-08-19 WO disclosed
US-20210147466-A1 IMPROVED PROCESSES FOR THE PREPARATION OF GUADECITABINE AND INTERMEDIATES THEREOF TEVA CZECH INDUSTRIES S.R.O. (CZ) 2021-05-20 US disclosed
CN-109071579-B Method for producing monomer for single-stranded nucleic acid molecule 住友化学株式会社 2021-05-14 CN disclosed
EP-3450439-B1 METHOD FOR PRODUCING MONOMER FOR SINGLE-STRANDED NUCLEIC ACID MOLECULE SUMITOMO CHEMICAL CO (JP) 2021-01-20 EP disclosed
EP-3634972-A2 IMPROVED PROCESSES FOR THE PREPARATION OF GUADECITABINE AND INTERMEDIATES THEREOF Teva Czech Industries s.r.o. (CZ) 2020-04-15 EP disclosed
US-20120202856-A1 SUBSTITUTED BENZIMDAZOLE DERIVATIVES USEFUL AS TRPM8 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2012-08-09 US disclosed
US-8217060-B2 Benzimidazole derivatives useful as TRP M8 receptor modulators JANSSEN PHARMACEUTICA, NV (BE) 2012-07-10 US disclosed
US-20110183974-A1 1,2,4-OXADIAZOLE SUBSTITUTED PIPERIDINE AND PIPERAZINE DERIVATIVES AS SMO ANTAGONISTS INSTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI (IT) 2011-07-28 US disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
US-7863294-B2 Heterocycle derivatives as histone deacetylase (HDAC) inhibitors INSTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-01-04 US disclosed
WO-2010132247-A1 BENZIMIDAZOLE DERIVATIVES USEFUL AS TRP M8 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2010-11-18 WO disclosed
US-20100292276-A1 BENZIMIDAZOLE DERIVATIVES USEFUL AS TRP M8 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, NV (BE) 2010-11-18 US disclosed
US-7320995-B2 Benzimidazoles and benzothiazoles as inhibitors of map kinase ELI LILLY AND COMPANY (US) 2008-01-22 US disclosed
US-20050272791-A1 Benzimidazoles and benzothiazoles as inhibitors of map kinase EIL LILLY AND COMPANY (US) 2005-12-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120202856-A1 SUBSTITUTED BENZIMDAZOLE DERIVATIVES USEFUL AS TRPM8 RECEPTOR MODULATORS TRPM8, TRPV1, TRPA1 RAB9A 2533/4885SMN1; SMN2 1255/4885HTT 4162/4885
US-20050272791-A1 Benzimidazoles and benzothiazoles as inhibitors of map kinase MAP3K8, MAPK8, MAPK1 RAB9A 1985/4885SMN1; SMN2 4631/4885HTT 4541/4885
US-20210147466-A1 IMPROVED PROCESSES FOR THE PREPARATION OF GUADECITABINE AND INTERMEDIATES THEREOF UNG, SAMHD1, ALKBH1 RAB9A 2077/4885SMN1; SMN2 960/4885HTT 2449/4885
US-20110183974-A1 1,2,4-OXADIAZOLE SUBSTITUTED PIPERIDINE AND PIPERAZINE DERIVATIVES AS SMO ANTAGONISTS SHH, SMO, GLI1 RAB9A 2234/4885SMN1; SMN2 518/4885HTT 3454/4885
US-20100292276-A1 BENZIMIDAZOLE DERIVATIVES USEFUL AS TRP M8 RECEPTOR MODULATORS TRPM8, TRPV1, TRPA1 RAB9A 2807/4885SMN1; SMN2 2716/4885HTT 2964/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.