SCHEMBL20366552

SCHEMBL20366552

COc1cc2c(cc1SN1CCCC1)CCC(=O)C2(C)C

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 2/20 0.34
PARP1 P09874 2/20 0.33
ALDH1A1 P00352 3/20 0.31
TSHR P16473 3/20 0.31
GAA P10253 2/20 0.31
NPBWR1 P48145 1/20 0.31
CHRM2 P08172 1/20 0.31
ADRA2A P08913 1/20 0.31
MAPK1 P28482 2/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HPGD P15428 2/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20004608 0.91 ALK (0.33) ALKPARP1ALDH1A1GAAMEN1
SCHEMBL20004650 0.81 ALK (0.38) ALKPARP1ALDH1A1MAPK1KMT2A
SCHEMBL897635 0.76 ALDH1A1 (0.58) ALDH1A1TSHRGAANPBWR1MEN1
SCHEMBL20004206 0.75 ALK (0.38) ALKPARP1ALDH1A1GAAMAPK1
SCHEMBL1755954 0.74 ALK (0.33) ALKPARP1
SCHEMBL897525 0.74 ALK (0.43) ALKALDH1A1TSHRGAAMAPK1
SCHEMBL897012 0.74 HTR2A (0.45) ALKTSHRKDM4E
SCHEMBL20061137 0.74 S100B (0.38) ALKPARP1ALDH1A1TSHRGAA
SCHEMBL29940534 0.73 ALK (0.38) ALKPARP1ALDH1A1TSHRGAA
SCHEMBL27087621 0.73 ALK (0.38) ALKPARP1ALDH1A1TSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3613729-A1 TETRACYCLIC COMPOUNDS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2020-02-26 EP disclosed
EP-3345903-B1 TETRACYCLIC COMPOUNDS CHUGAI PHARMACEUTICAL CO LTD (JP) 2019-10-09 EP disclosed
EP-3345903-A1 TETRACYCLIC COMPOUNDS Chugai Seiyaku Kabushiki Kaisha (JP) 2018-07-11 EP disclosed