SCHEMBL203904

SCHEMBL203904

CC(C)(C)OC(=O)N[C@@H]1CCCNC1=O

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 14/20 0.60
GAA P10253 1/20 0.55
CCR1 P32246 1/20 0.48
CCR5 P51681 1/20 0.48
CXCR4 P61073 1/20 0.48
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2462209 1.00 CCR2 (0.60) CCR2GAACCR1CCR5CXCR4
SCHEMBL2460843 1.00 CCR2 (0.60) CCR2GAACCR1CCR5CXCR4
SCHEMBL203905 1.00 CCR2 (0.60) CCR2GAACCR1CCR5CXCR4
SCHEMBL29418355 1.00 CCR2 (0.60) CCR2GAACCR1CCR5CXCR4
SCHEMBL2329779 0.95 CCR2 (0.67) CCR2GAACCR1CCR5CXCR4
SCHEMBL4704983 0.95 CCR2 (0.67) CCR2GAACCR1CCR5CXCR4
SCHEMBL2462379 0.95 CCR2 (0.67) CCR2GAACCR1CCR5CXCR4
SCHEMBL7327118 0.93 CCR2 (0.57) CCR2GAACCR1CCR5CXCR4
SCHEMBL7327122 0.93 CCR2 (0.57) CCR2GAACCR1CCR5CXCR4
Acetic Acid SCHEMBL8778037 0.92 CCR2 (0.62) CCR2GAACCR1CCR5CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4644380-A1 PYRIDAZINE NLRP3 INHIBITOR COMPOUND, PHARMACEUTICAL COMPOSITION, AND PREPARATION METHOD THEREFOR AND USE THEREOF Changchun Genescience Pharmaceutical Co., Ltd. (CN) 2025-11-05 EP disclosed
CN-115916207-A Five-membered and six-membered heterocyclic compounds and application thereof as protein receptor kinase inhibitors 轶诺(浙江)药业有限公司 2023-04-04 CN disclosed
US-11530183-B2 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists BRISTOL-MYERS SQUIBB COMPANY (US) 2022-12-20 US disclosed
CN-106588890-B Antiviral compounds 吉利德制药有限责任公司 2020-11-27 CN disclosed
EP-3626716-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2020-03-25 EP disclosed
US-9981955-B2 Antiviral compounds GILEAD PHARMASSET LLC (US) 2018-05-29 US disclosed
EP-3309157-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2018-04-18 EP disclosed
EP-3002281-B1 ANTIVIRAL COMPOUNDS GILEAD PHARMASSET LLC (US) 2017-09-13 EP disclosed
US-20170029408-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. 2017-02-02 US disclosed
US-9511056-B2 Antiviral compounds GILEAD PHARMASSET LLC (US) 2016-12-06 US disclosed
US-20120157404-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2012-06-21 US disclosed
US-8088368-B2 Antiviral compounds GILEAD SCIENCES, INC. (US) 2012-01-03 US disclosed
WO-2011117160-A1 PYRROLOPYRAZINE DERIVATIVES AND THEIR USE AS JAK AND SYK INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2011-09-29 WO disclosed
US-20110230414-A1 Pyrrolopyrazine Kinase Inhibitors HENDRICKS ROBERT THAN 2011-09-22 US disclosed
CN-101270076-B Method for preparing natural product (3S,9S)-Ciliatamides C UNIV FUDAN 2011-04-27 CN disclosed
US-20100310512-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. 2010-12-09 US disclosed
US-7531657-B2 Method for preparing sulphostin and analogue thereof or preparation intermediate thereof NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2009-05-12 US disclosed
CN-101270076-A Method for preparing natural product (3S,9S)-Ciliatamides C UNIV FUDAN (CN) 2008-09-24 CN disclosed
US-20050020834-A1 Method for preparation of sulphostin and its analogue or intermediates thereof NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2005-01-27 US disclosed
EP-1457494-A1 PROCESSES FOR PREPARATION OF SULPHOSTIN AND ITS ANALOGUES OR INTERMEDIATES THEREOF Nippon Kayaku Kabushiki Kaisha (JP) 2004-09-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050020834-A1 Method for preparation of sulphostin and its analogue or intermediates thereof SOST, PTMS, FGF23 CCR2 1659/4885GAA 2919/4885CCR1 930/4885
US-20170029408-A1 ANTIVIRAL COMPOUNDS MAVS, EIF2AK2, ZC3HAV1 CCR2 1607/4885GAA 151/4885CCR1 795/4885
US-20120157404-A1 ANTIVIRAL COMPOUNDS MAVS, EIF2AK2, ZC3HAV1 CCR2 1607/4885GAA 151/4885CCR1 795/4885
US-11530183-B2 Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists FPR1, FPR2, FPR3 CCR2 13/4885GAA 4579/4885CCR1 81/4885
US-20110230414-A1 Pyrrolopyrazine Kinase Inhibitors SYK, ZAP70, JAK2 CCR2 1035/4885GAA 3087/4885CCR1 2908/4885
US-20100310512-A1 ANTIVIRAL COMPOUNDS MAVS, EIF2AK2, ZC3HAV1 CCR2 1607/4885GAA 151/4885CCR1 795/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.