SCHEMBL2053324

SCHEMBL2053324

Fc1cccc(F)c1-c1[c]ccc(C(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.38
F7 P08709 1/20 0.38
F3 P13726 1/20 0.38
TSHR P16473 2/20 0.37
MAPK1 P28482 1/20 0.37
MAT2A P31153 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
PDE2A O00408 3/20 0.36
MGLL Q99685 1/20 0.34
P2RX1 P51575 1/20 0.34
P2RX7 Q99572 1/20 0.34
ALDH1A1 P00352 2/20 0.32
LMNA P02545 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
IDO1 P14902 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2049535 0.81 HSD11B1 (0.35) CES2TSHRMAPK1MAT2ATAAR1
SCHEMBL2432403 0.81 GPR3 (0.41) CES2TSHRMAT2APDE2AALDH1A1
SCHEMBL2050518 0.78 L3MBTL1 (0.37) PDE2AALDH1A1L3MBTL1
SCHEMBL2204411 0.76 NOTUM (0.43) CES2TSHRMAPK1MGLLIDO1
SCHEMBL2431003 0.76 PTPN1 (0.39) CES2TSHRMAPK1MAT2ATAAR1
SCHEMBL1370057 0.74 KIF11 (0.47) CES2TSHRMAPK1ALDH1A1L3MBTL1
SCHEMBL2049079 0.74 ACHE (0.39) MAPK1ALDH1A1
SCHEMBL2015248 0.74 TRPA1 (0.43) PDE2AIDO1
SCHEMBL1690372 0.73 SMN1; SMN2 (0.34) CES2MAPK1PDE2ALMNA
SCHEMBL2013705 0.73 RXRA (0.33) CES2TSHRMAPK1PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed