SCHEMBL21088883

SCHEMBL21088883

O=C(O)CCN1CCC2(CC1)CC(NC1CC1)C2

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 7/20 0.44
ITGB3 P05106 7/20 0.41
ITGA2B P08514 7/20 0.41
GLA P06280 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.34
CYP1A2 P05177 1/20 0.34
MAPK1 P28482 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33
APEX1 P27695 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25924012 0.87 L3MBTL1 (0.45) KDM1AITGB3ITGA2BSMN1; SMN2MAPK1
SCHEMBL21088777 0.84 KDM1A (0.40) KDM1AITGB3ITGA2BGLAAPEX1
SCHEMBL25923906 0.81 KDM1A (0.46) KDM1ASMN1; SMN2
SCHEMBL21088467 0.80 CNR1 (0.37) KDM1ASMN1; SMN2
SCHEMBL25923937 0.78 KDM1A (0.40) KDM1ACYP1A2
SCHEMBL21088867 0.75 HTR4 (0.35) KDM1A
SCHEMBL29326474 0.75 ITGB3 (0.43) KDM1AITGB3ITGA2BGLASMN1; SMN2
SCHEMBL25923925 0.74 KDM1A (0.42) KDM1ACYP1A2
SCHEMBL25924008 0.74 KDM1A (0.32) KDM1A
SCHEMBL21088586 0.73 KDM1A (0.31) KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286172-B1 LSD1 INHIBITORS AND USES THEREOF CONSTELLATION PHARMACEUTICALS INC (US) 2019-06-12 EP disclosed